Y-27632

Y-27632

SCHEMBL28416532

CC(N)[C@H]1CC[C@@H](C(=O)Nc2ccncc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 8/20 1.00
ROCK1 Q13464 8/20 1.00
PKN2 Q16513 4/20 1.00
RPS6KA5 O75582 3/20 1.00
LRRK2 Q5S007 3/20 1.00
TP53 P04637 2/20 1.00
CYP3A4 P08684 2/20 1.00
PRKD3 O94806 2/20 1.00
CDK1 P06493 2/20 1.00
CDK2 P24941 2/20 1.00
LTK P29376 2/20 1.00
CDK8 P49336 2/20 1.00
PRKX P51817 2/20 1.00
PRKCQ Q04759 2/20 1.00
PRKCD Q05655 2/20 1.00
STK3 Q13188 2/20 1.00
CDC42BPA Q5VT25 2/20 1.00
BRSK1 Q8TDC3 2/20 1.00
CLK4 Q9HAZ1 2/20 1.00
TSHR P16473 2/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Y-27632 SCHEMBL598993 1.00 ROCK2 (1.00) ROCK2ROCK1PKN2RPS6KA5LRRK2
Y-27632 SCHEMBL190356 1.00 ROCK2 (1.00) ROCK2ROCK1PKN2RPS6KA5LRRK2
Y-27632 SCHEMBL1980406 1.00 ROCK2 (1.00) ROCK2ROCK1PKN2RPS6KA5LRRK2
Y-27632 SCHEMBL20333114 1.00 ROCK2 (1.00) ROCK2ROCK1PKN2RPS6KA5LRRK2
Y-27632 SCHEMBL18935698 1.00 ROCK2 (1.00) ROCK2ROCK1PKN2RPS6KA5LRRK2
Y-27632 SCHEMBL342816 1.00 ROCK2 (1.00) ROCK2ROCK1PKN2RPS6KA5LRRK2
Y-27632 SCHEMBL30286315 1.00 ROCK2 (1.00) ROCK2ROCK1PKN2RPS6KA5LRRK2
Y-27632 SCHEMBL2796890 0.99 ROCK2 (0.97) ROCK2ROCK1PKN2RPS6KA5LRRK2
Y-27632 SCHEMBL1554110 0.99 ROCK2 (1.00) ROCK2ROCK1PKN2RPS6KA5LRRK2
Y-27632 SCHEMBL2834049 0.99 ROCK2 (1.00) ROCK2ROCK1PKN2RPS6KA5LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113015429-A Method and container for preserving corneal endothelial cells 学校法人同志社 2021-06-22 CN disclosed
CN-107082747-B Compounds for targeted drug delivery and enhancing siRNA activity 日东电工株式会社 2020-11-20 CN disclosed
CN-107043334-B Compounds for targeted drug delivery and enhancing siRNA activity 日东电工株式会社 2020-06-16 CN disclosed