SCHEMBL28439331

SCHEMBL28439331

CCCCCCCCCCn1cc(N)cc(N)c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.41
PTGS2 P35354 3/20 0.41
MGLL Q99685 2/20 0.41
FAAH O00519 1/20 0.41
TLR8 Q9NR97 5/20 0.40
CYP1A2 P05177 3/20 0.39
CYP2C19 P33261 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
GAA P10253 1/20 0.39
MEN1 O00255 1/20 0.39
CYP2C9 P11712 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 1/20 0.38
GPR84 Q9NQS5 1/20 0.37
TYR P14679 1/20 0.37
CYP19A1 P11511 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28440804 1.00 PTGS1 (0.41) PTGS1PTGS2MGLLFAAHTLR8
SCHEMBL28435216 1.00 PTGS1 (0.41) PTGS1PTGS2MGLLFAAHTLR8
SCHEMBL11449602 0.77 AURKA (0.59) TLR8CYP1A2CYP2C19MEN1CYP2C9
SCHEMBL16812286 0.77 TYR (0.41) TLR8TDP1TYRNPC1L3MBTL1
SCHEMBL7196320 0.73 ADORA2B (0.49) PTGS1PTGS2MGLLFAAHTLR8
SCHEMBL18161040 0.72 TYR (0.38) TLR8CYP1A2CYP2C19CYP2C9ALDH1A1
SCHEMBL4146972 0.71 ADORA2B (0.40) PTGS1PTGS2MGLLFAAHTLR8
SCHEMBL2215259 0.70 CYP1A2 (0.60) TLR8CYP1A2CYP2C19TDP1GAA
SCHEMBL4685541 0.70 TDP1 (0.41) PTGS1PTGS2MGLLFAAHTLR8
SCHEMBL4156451 0.68 PDE4A (0.43) TDP1TYRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111533741-B Macrocyclic compound with hydrophobic inner cavity and preparation method thereof 江南大学 2021-04-30 CN disclosed
CN-111533741-A Macrocyclic compound with hydrophobic inner cavity and preparation method thereof 江南大学 2020-08-14 CN disclosed