SCHEMBL2844641

SCHEMBL2844641

O=C(O)NCCCc1ccnc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
LOXL2 Q9Y4K0 1/20 0.46
CASP1 P29466 1/20 0.45
HTR1A P08908 2/20 0.44
ADRA1D P25100 2/20 0.44
ADRA1A P35348 2/20 0.44
ADRA1B P35368 2/20 0.44
NSD2 O96028 1/20 0.44
FAAH O00519 1/20 0.43
MTNR1A P48039 7/20 0.43
MTNR1B P49286 7/20 0.43
FLT1 P17948 1/20 0.41
KDR P35968 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2846544 0.96 CYP1A2 (0.48) CYP1A2LOXL2CASP1HTR1AADRA1D
SCHEMBL2841416 0.94 HTR1A (0.49) CYP1A2LOXL2CASP1HTR1AADRA1D
SCHEMBL2937018 0.81 CYP1A2 (0.54) CYP1A2LOXL2HTR1AADRA1DADRA1A
SCHEMBL10243391 0.81 CASP1 (0.45) CASP1MTNR1AMTNR1BFLT1KDR
SCHEMBL20562641 0.81 CASP1 (0.53) CASP1NSD2MTNR1AMTNR1B
SCHEMBL5273635 0.80 CYP1A2 (0.52) CYP1A2LOXL2CASP1ADRA1AFAAH
SCHEMBL12304975 0.79 NAMPT (0.49) CASP1MTNR1AMTNR1BTSHR
SCHEMBL2408804 0.79 LOXL2 (0.41) CYP1A2LOXL2CASP1HTR1AADRA1D
SCHEMBL5210378 0.79 CYP1A2 (0.51) CYP1A2LOXL2ADRA1A
SCHEMBL7832661 0.78 MAPT (0.51) CYP1A2LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2251324-A1 HETEROARYL-ALKYLCARBAMATE COMPOUNDS AND THEIR USE AS INHIBITORS OF THE FAAH ENZYME Sanofi-Aventis (FR) 2010-11-17 EP disclosed
EP-1720829-B1 DERIVATIVES OF HETEROARYL-ALKYLCARBAMATES, PREPARATION METHOD THEREOF AND USE OF SAME AS FAAH ENZYME INHIBITORS SANOFI AVENTIS (FR) 2009-10-14 EP disclosed