SCHEMBL28456589

SCHEMBL28456589

CC(C)[Si](N[Si](c1ccccc1)(C(C)C)C(C)C)(c1ccccc1)C(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.39
AOC3 Q16853 1/20 0.37
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
CYP19A1 P11511 1/20 0.34
TAAR1 Q96RJ0 4/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
GAA P10253 2/20 0.33
ATM Q13315 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP3A4 P08684 2/20 0.33
ALOX15 P16050 2/20 0.33
TSHR P16473 2/20 0.33
ALOX12 P18054 2/20 0.33
HSD17B10 Q99714 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
THRB P10828 1/20 0.33
RECQL P46063 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2267663 0.85 TDP1 (0.36) TDP1AOC3ESR1ESR2TAAR1
SCHEMBL2269102 0.81 SIGMAR1 (0.39) TDP1AOC3TAAR1GAAMEN1
SCHEMBL705725 0.74 ESR1 (0.34) TDP1AOC3ESR1ESR2CYP19A1
SCHEMBL705425 0.74 ESR1 (0.34) TDP1AOC3ESR1ESR2CYP19A1
SCHEMBL706818 0.74 MAOA (0.36) TDP1AOC3ESR1ESR2TAAR1
SCHEMBL13766348 0.72 ESR1 (0.37) TDP1ESR1ESR2CYP19A1TAAR1
SCHEMBL5180601 0.72 ESR1 (0.37) TDP1ESR1ESR2CYP19A1TAAR1
SCHEMBL9763717 0.72 ESR1 (0.37) TDP1ESR1ESR2CYP19A1TAAR1
SCHEMBL985723 0.72 ESR1 (0.37) TDP1ESR1ESR2CYP19A1TAAR1
SCHEMBL1316040 0.72 ESR1 (0.38) TDP1AOC3ESR1ESR2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107964016-B Thiophene derivatives 天津合美医药科技有限公司 2021-10-01 CN disclosed
CN-108059635-B Thiophene derivatives 天津合美医药科技有限公司 2021-10-01 CN disclosed
CN-107722036-B Thiophene derivatives 天津合美医药科技有限公司 2020-09-04 CN disclosed