SCHEMBL28461597

SCHEMBL28461597

COc1cccc(-c2ccc3cn(C4CCCN(C(=O)OC(C)(C)C)C4)nc3c2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.50
SRC P12931 2/20 0.50
ABL1 P00519 1/20 0.50
ABL2 P42684 1/20 0.50
USP30 Q70CQ3 2/20 0.45
GRM5 P41594 1/20 0.42
NPC1 O15118 4/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
FGFR3 P22607 1/20 0.41
KDR P35968 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
CRHBP P24387 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
CRHR2 Q13324 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28458581 0.92 SRC (0.47) EGFRSRCABL1ABL2USP30
SCHEMBL28460213 0.89 USP30 (0.45) EGFRSRCABL1ABL2USP30
SCHEMBL28452589 0.89 USP30 (0.45) EGFRSRCABL1ABL2USP30
SCHEMBL28458345 0.86 BTK (0.45) EGFRSRCABL1ABL2USP30
SCHEMBL28458448 0.86 GPR119 (0.48) ABL1USP30FGFR3KDRCHEK2
SCHEMBL28898133 0.86 APLNR (0.44) EGFRSRCABL1ABL2USP30
SCHEMBL29968466 0.86 GPR119 (0.48) ABL1USP30FGFR3KDRCHEK2
SCHEMBL28449733 0.86 CNR1 (0.46) USP30MEN1KMT2ACHEK2BTK
SCHEMBL28461486 0.86 GPR119 (0.46) USP30FGFR3KDRCHEK2
SCHEMBL28898963 0.86 HDAC1 (0.46) USP30FGFR3KDRCHEK2IRAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662232-B Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2022-08-02 CN disclosed
CN-111662232-A Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2020-09-15 CN disclosed