SCHEMBL28463141

SCHEMBL28463141

O=C(Nc1ccccc1S)c1cc(Cl)c(O)c(Cl)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.65
MDM4 O15151 4/20 0.65
MDM2 Q00987 2/20 0.65
TOP1 P11387 2/20 0.54
TOP2A P11388 1/20 0.54
TOP2B Q02880 1/20 0.54
HSD17B13 Q7Z5P4 3/20 0.53
TAS1R3 Q7RTX0 1/20 0.49
TAS1R1 Q7RTX1 1/20 0.49
TAS1R2 Q8TE23 1/20 0.49
ALDH1A1 P00352 4/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
LMNA P02545 2/20 0.47
HPGD P15428 2/20 0.47
HTT P42858 1/20 0.47
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11588151 0.84 NPC1 (0.66) TP53TOP1TOP2ATOP2BHSD17B13
SCHEMBL31312812 0.82 TAS1R3 (0.73) TP53MDM4MDM2TAS1R3TAS1R1
SCHEMBL25349072 0.81 RAB9A (0.64) TOP1TOP2ATOP2BHSD17B13TAS1R3
SCHEMBL333488 0.78 MDM4 (1.00) TP53MDM4MDM2MEN1KMT2A
SCHEMBL6002243 0.76 MDM4 (0.96) TP53MDM4MDM2MEN1KMT2A
SCHEMBL14890169 0.76 CYP1A2 (0.74) TP53MDM4MDM2ALDH1A1LMNA
SCHEMBL11589239 0.75 NPC1 (0.57) TP53TOP1TOP2ATOP2BHSD17B13
SCHEMBL11589478 0.74 MEN1 (0.56) TP53TOP1TOP2ATOP2BHSD17B13
SCHEMBL11588024 0.73 HSD17B13 (0.48) TP53TOP1TOP2ATOP2BHSD17B13
SCHEMBL1520421 0.72 MEN1 (0.77) TP53MDM4MDM2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111793039-A Preparation method of dortinode 苏州明锐医药科技有限公司 2020-10-20 CN claimed
CN-111675675-A Preparation method of dortinode 苏州明锐医药科技有限公司 2020-09-18 CN claimed