SCHEMBL28470683

SCHEMBL28470683

Cc1ccc(C#CC(=O)Cc2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCP P55072 1/20 0.54
FFAR1 O14842 3/20 0.50
L3MBTL1 Q9Y468 2/20 0.49
TDP1 Q9NUW8 1/20 0.49
KMT2A Q03164 3/20 0.48
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
PSMB8 P28062 1/20 0.43
PSMB5 P28074 1/20 0.43
MEN1 O00255 2/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
AKR1B1 P15121 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HSP90AA1 P07900 1/20 0.41
AGTR1 P30556 1/20 0.41
PAX8 Q06710 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28704543 0.93 VCP (0.58) VCPFFAR1L3MBTL1TDP1KMT2A
SCHEMBL28479005 0.88 FFAR1 (0.58) VCPFFAR1L3MBTL1KMT2AMEN1
SCHEMBL28480057 0.83 L3MBTL1 (0.57) FFAR1L3MBTL1TDP1KMT2ACNR2
SCHEMBL28824705 0.83 FFAR1 (0.50) FFAR1L3MBTL1CNR2SMN1; SMN2NPC1
SCHEMBL28754059 0.83 RAB9A (0.54) FFAR1L3MBTL1TDP1KMT2ACNR2
SCHEMBL29162927 0.83 FFAR1 (0.52) VCPFFAR1L3MBTL1NPC1RAB9A
SCHEMBL28704538 0.77 FFAR1 (0.54) FFAR1L3MBTL1CNR2NPC1RAB9A
SCHEMBL28689949 0.77 FFAR1 (0.54) FFAR1L3MBTL1KMT2ACNR1CNR2
SCHEMBL28685979 0.77 FFAR1 (0.54) FFAR1L3MBTL1TDP1KMT2ACNR1
SCHEMBL28824698 0.76 NPC1 (0.57) FFAR1L3MBTL1TDP1KMT2ACNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111892597-B Quinoxalinyl pyridopyrazine compound and preparation method and application thereof 山西天宏达安医药科技有限公司 2023-07-25 CN claimed
CN-111892597-A Quinoxalinyl pyridopyrazine compound and preparation method and application thereof 朱继强 2020-11-06 CN claimed
CN-111892597-B Quinoxalinyl pyridopyrazine compound and preparation method and application thereof 山西天宏达安医药科技有限公司 2023-07-25 CN disclosed
CN-110698426-B Method for preparing 1, 3-benzothiazole derivative by efficient catalysis of potassium tert-butoxide 陕西师范大学 2022-08-23 CN disclosed
CN-111892597-A Quinoxalinyl pyridopyrazine compound and preparation method and application thereof 朱继强 2020-11-06 CN disclosed
CN-110698426-A Method for preparing 1, 3-benzothiazole derivative by efficient catalysis of potassium tert-butoxide 陕西师范大学 2020-01-17 CN disclosed