SCHEMBL2849153

SCHEMBL2849153

O=C(Nc1ccncc1)c1cnn(-c2ccc(OC(F)(F)F)cc2)c1C(F)(F)F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.56
MET P08581 1/20 0.55
AXL P30530 1/20 0.55
MALT1 Q9UDY8 2/20 0.52
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
TRPC1 P48995 1/20 0.48
TRPC3 Q13507 1/20 0.48
STIM1 Q13586 1/20 0.48
ORAI1 Q96D31 1/20 0.48
STIM2 Q9P246 1/20 0.48
KDR P35968 3/20 0.48
FLT1 P17948 2/20 0.48
TRPV1 Q8NER1 1/20 0.47
NR3C1 P04150 2/20 0.46
LMNA P02545 1/20 0.46
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2855512 0.85 MALT1 (0.55) MAPTMETAXLMALT1KDM4E
SCHEMBL2852073 0.83 MAPT (0.71) MAPTMETAXLKDM4EALDH1A1
SCHEMBL2855275 0.83 MAPT (0.45) MAPTMETAXLKDM4ENPC1
SCHEMBL2856272 0.81 MALT1 (0.53) METAXLMALT1KDM4EALDH1A1
SCHEMBL2856196 0.80 MAPT (0.70) MAPTKDM4EALDH1A1NPC1RAB9A
SCHEMBL2850397 0.78 MALT1 (0.57) MAPTMETAXLMALT1KDM4E
SCHEMBL2850244 0.78 MALT1 (0.51) MAPTMETAXLMALT1KDM4E
SCHEMBL2858127 0.78 ALDH1A1 (0.74) MAPTMETAXLKDM4EALDH1A1
SCHEMBL21929518 0.76 NPC1 (0.55) MAPTMETAXLKDM4EALDH1A1
SCHEMBL2855560 0.76 ALDH1A1 (0.49) MAPTMETAXLKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed