SCHEMBL2850211

SCHEMBL2850211

CC(C)N(CCc1ccccc1)C(=O)c1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.49
POLB P06746 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
CCR1 P32246 3/20 0.44
HSP90AA1 P07900 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
MAPK1 P28482 1/20 0.43
GPR6 P46095 1/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
GRIA2 P42262 1/20 0.41
KEAP1 Q14145 2/20 0.40
NFE2L2 Q16236 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2862087 0.88 MAPT (0.51) MAPTPOLBSMN1; SMN2ALDH1A1KDM4E
SCHEMBL2854529 0.85 MAPT (0.47) MAPTPOLBSMN1; SMN2ALDH1A1KDM4E
SCHEMBL2854321 0.82 MAPT (0.53) MAPTPOLBSMN1; SMN2ALDH1A1KDM4E
SCHEMBL2854667 0.80 ALDH1A1 (0.55) MAPTPOLBSMN1; SMN2ALDH1A1KDM4E
SCHEMBL2853014 0.78 KDM4E (0.60) MAPTPOLBSMN1; SMN2ALDH1A1KDM4E
SCHEMBL2857362 0.77 ALDH1A1 (0.49) MAPTPOLBSMN1; SMN2ALDH1A1KDM4E
SCHEMBL2854414 0.77 MAPT (0.53) MAPTPOLBSMN1; SMN2ALDH1A1KDM4E
SCHEMBL10366449 0.77 MAPT (0.53) MAPTPOLBSMN1; SMN2ALDH1A1KDM4E
SCHEMBL2855694 0.75 MAPK14 (0.49) MAPTALDH1A1HSP90AA1NPSR1MAPK1
SCHEMBL2852015 0.75 CCR1 (0.63) MAPTPOLBSMN1; SMN2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed