SCHEMBL28503293

SCHEMBL28503293

O=C(O)CCOc1nc2ccccc2c(=O)[nH]1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.59
PARP2 Q9UGN5 1/20 0.59
MAPK1 P28482 1/20 0.56
HCAR2 Q8TDS4 2/20 0.49
KDM4C Q9H3R0 1/20 0.49
RAB9A P51151 1/20 0.49
MMP13 P45452 1/20 0.48
CYP1B1 Q16678 1/20 0.48
MAPT P10636 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
MAOB P27338 2/20 0.47
TNKS2 Q9H2K2 3/20 0.47
QTRT1 Q9BXR0 1/20 0.46
KMT2A Q03164 1/20 0.46
TNKS O95271 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
LMNA P02545 1/20 0.44
PKM P14618 1/20 0.44
GUSB P08236 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28502323 0.84 HCAR2 (0.53) PARP1PARP2HCAR2KDM4CRAB9A
SCHEMBL6886533 0.82 TNKS2 (0.56) PARP1HCAR2KDM4CRAB9AMAOB
SCHEMBL6004217 0.81 TNKS2 (0.51) PARP1HCAR2KDM4CRAB9AMAOB
Hydrochloric Acid SCHEMBL15742407 0.78 KDM4C (0.65) PARP1KDM4CRAB9ATNKS2QTRT1
SCHEMBL6473755 0.78 KDM4C (0.75) PARP1HCAR2KDM4CRAB9AMAOB
SCHEMBL23068618 0.76 PARP1 (0.59) PARP1PARP2TNKS2TNKS
SCHEMBL6597891 0.76 ACHE (0.48) PARP1HCAR2KDM4CRAB9AMAOB
SCHEMBL2718160 0.75 PARP1 (1.00) PARP1PARP2MAPTTNKS2KMT2A
SCHEMBL29903052 0.75 PARP1 (1.00) PARP1PARP2MAPTTNKS2KMT2A
SCHEMBL38651228 0.74 HTR3A (0.56) PARP1PARP2MAPTTNKS2TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107226808-B Tankyrase inhibitors 北京四环制药有限公司 2021-01-01 CN disclosed