SCHEMBL28506409

SCHEMBL28506409

CN1CCC(N(C)C(=O)c2ccc(B(O)O)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.48
LMNA P02545 2/20 0.48
CCR5 P51681 2/20 0.46
PDK2 Q15119 2/20 0.45
HRH3 Q9Y5N1 1/20 0.45
ALDH1A1 P00352 1/20 0.44
BRD4 O60885 1/20 0.44
TAF1 P21675 1/20 0.44
CECR2 Q9BXF3 1/20 0.44
USP30 Q70CQ3 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
TLR9 Q9NR96 1/20 0.43
TLR8 Q9NR97 1/20 0.43
TLR7 Q9NYK1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28506326 0.92 MCHR1 (0.58) MCHR1CCR5HRH3USP30
SCHEMBL949827 0.88 ALDH1A1 (0.46) LMNACCR5PDK2ALDH1A1BRD4
SCHEMBL29954467 0.84 ALDH1A1 (0.56) LMNAALDH1A1BRD4
SCHEMBL25498560 0.84 LMNA (0.65) MCHR1LMNACCR5PDK2HRH3
SCHEMBL12082859 0.84 PDK2 (0.61) MCHR1LMNACCR5PDK2HRH3
SCHEMBL16553814 0.82 HTR2A (0.54) MCHR1LMNACCR5PDK2HRH3
SCHEMBL1164100 0.82 MCHR1 (0.50) MCHR1LMNACCR5PDK2HRH3
SCHEMBL94337 0.82 MCHR1 (0.50) MCHR1LMNACCR5PDK2HRH3
SCHEMBL3329900 0.82 CCR5 (0.55) MCHR1CCR5HRH3USP30ADORA2A
SCHEMBL21077844 0.80 MCHR1 (0.58) MCHR1LMNACCR5PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed