SCHEMBL28508255

SCHEMBL28508255

O=C(c1ccc2nc(-c3ccccc3)n(Cc3ccccc3)c2c1)N1CCOCC1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 7/20 0.52
HRH3 Q9Y5N1 6/20 0.52
ALDH1A1 P00352 3/20 0.51
PDE6D O43924 1/20 0.51
ALDH2 P05091 1/20 0.51
ALDH3A1 P30838 1/20 0.51
HTT P42858 1/20 0.49
PKM P14618 2/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28507437 0.92 PTGER4 (0.55) HRH3ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL28503579 0.82 ALDH1A1 (0.63) BRD4ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL28503584 0.82 PIK3CA (0.62) ALDH1A1CYP2C19
SCHEMBL22955650 0.80 AGTR1 (0.48) ALDH1A1PKMNPC1RAB9A
SCHEMBL22955584 0.80 HTR2C (0.45) ALDH1A1CYP2C9CYP2C19
SCHEMBL28505411 0.77 DRD2 (0.66) BRD4ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL22955374 0.77 HTR2C (0.48)
SCHEMBL22955902 0.76 HTR2C (0.44) PKMNPC1RAB9A
SCHEMBL14382294 0.76 PDE2A (0.61) BRD4ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL20467484 0.74 HPGD (0.77) ALDH1A1HTTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107311933-B Benzimidazole derivative, preparation method and application thereof 中国人民解放军军事医学科学院毒物药物研究所 2020-12-22 CN disclosed