SCHEMBL28503584

SCHEMBL28503584

O=C(NCCN1CCOCC1)c1ccc2nc(-c3ccccc3)n(Cc3ccccc3)c2c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.62
HPGD P15428 3/20 0.59
CD274 Q9NZQ7 1/20 0.59
KMT2A Q03164 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C19 P33261 1/20 0.57
PDE2A O00408 1/20 0.56
KDM4E B2RXH2 3/20 0.55
MAPT P10636 1/20 0.55
ATM Q13315 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
ALDH1A1 P00352 2/20 0.54
GAA P10253 2/20 0.54
GLA P06280 1/20 0.54
HSD17B10 Q99714 1/20 0.54
PTGER4 P35408 2/20 0.53
POLB P06746 1/20 0.53
MEN1 O00255 1/20 0.52
AGTR1 P30556 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28508255 0.82 BRD4 (0.52) CYP2C19ALDH1A1
SCHEMBL28507636 0.80 ACSS2 (0.59) PDE2AALDH1A1PTGER4
SCHEMBL28503586 0.79 BRD4 (0.51) PDE2AALDH1A1
SCHEMBL28514126 0.79 PDE6D (0.47) PIK3CAHPGDPDE2AKDM4EALDH1A1
SCHEMBL28510597 0.78 ACSS2 (0.61)
SCHEMBL28513264 0.78 TP53 (0.53) PDE2AMAPTALDH1A1GAAPOLB
SCHEMBL28516171 0.78 THRB (0.50) PDE2AMAPTALDH1A1
SCHEMBL2162541 0.78 KMT2A (0.90) PIK3CAKMT2AMAPTPOLBMEN1
SCHEMBL28503579 0.77 ALDH1A1 (0.63) HPGDKDM4EMAPTALDH1A1HSD17B10
SCHEMBL28510581 0.76 SMN1; SMN2 (0.59) PDE2AMAPTPTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107311933-B Benzimidazole derivative, preparation method and application thereof 中国人民解放军军事医学科学院毒物药物研究所 2020-12-22 CN disclosed