SCHEMBL28510033

SCHEMBL28510033

O=C(NN=Cc1ccc(O)c(O)c1)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX4 Q9NPH5 1/20 0.79
MAPT P10636 8/20 0.77
GAA P10253 3/20 0.77
POLB P06746 2/20 0.77
LMNA P02545 3/20 0.69
DUSP3 P51452 2/20 0.69
PTPN5 P54829 2/20 0.69
PTPN11 Q06124 2/20 0.69
SMN1; SMN2 Q16637 1/20 0.69
L3MBTL1 Q9Y468 1/20 0.69
ALDH1A1 P00352 2/20 0.69
NPSR1 Q6W5P4 2/20 0.69
SENP1 Q9P0U3 1/20 0.69
KMT2A Q03164 3/20 0.68
MEN1 O00255 2/20 0.68
RAB9A P51151 1/20 0.68
GFER P55789 2/20 0.66
HTT P42858 2/20 0.64
KDM4E B2RXH2 1/20 0.64
AGTR1 P30556 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8298517 1.00 NOX4 (0.79) NOX4MAPTGAAPOLBLMNA
SCHEMBL28510030 0.88 LMNA (0.76) MAPTGAAPOLBLMNADUSP3
SCHEMBL28517560 0.87 MAPT (1.00) MAPTGAAPOLBLMNADUSP3
SCHEMBL28515477 0.87 MAPT (1.00) MAPTGAAPOLBLMNADUSP3
SCHEMBL28512241 0.87 MAPT (0.84) MAPTGAAPOLBLMNADUSP3
SCHEMBL21292850 0.84 DUSP3 (0.82) MAPTGAAPOLBLMNADUSP3
SCHEMBL21292847 0.84 DUSP3 (0.82) MAPTGAAPOLBLMNADUSP3
SCHEMBL28528683 0.84 MAPT (0.80) MAPTGAAPOLBLMNADUSP3
SCHEMBL2663942 0.83 MAPT (0.69) MAPTGAAPOLBLMNADUSP3
SCHEMBL15917497 0.83 MAPT (0.80) MAPTGAAPOLBLMNADUSP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112079744-A Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2020-12-15 CN claimed
CN-112079744-B Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2021-07-30 CN disclosed
CN-112079744-A Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2020-12-15 CN disclosed