SCHEMBL28510375

SCHEMBL28510375

O=C(Cc1ccccc1)ONS(=O)(=O)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.48
ERBB2 P04626 5/20 0.48
ALDH1A1 P00352 2/20 0.47
MAPK1 P28482 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
KEAP1 Q14145 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
PAM P19021 1/20 0.46
TSHR P16473 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
MMP1 P03956 1/20 0.44
MMP2 P08253 1/20 0.44
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44
MMP13 P45452 1/20 0.44
PRMT1 Q99873 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8707459 0.81 ALDH1A1 (0.53) ALDH1A1MAPK1HDAC1HDAC8PRMT1
SCHEMBL27445747 0.81 TSHR (0.50) ALDH1A1MAPK1L3MBTL1HDAC8PAM
SCHEMBL7053278 0.81 BCAT1 (0.46) EGFRERBB2ALDH1A1TSHRCA1
SCHEMBL1925760 0.80 POLB (0.56) EGFRERBB2ALDH1A1MAPK1L3MBTL1
SCHEMBL28424543 0.80 ADAMTS4 (0.54) MAPK1TSHRMMP1MMP2MMP9
SCHEMBL10687684 0.79 ALDH1A1 (0.45) ALDH1A1TSHRCA1CA2MMP1
SCHEMBL28745516 0.78 MMP12 (0.53) ALDH1A1L3MBTL1KEAP1HDAC1TSHR
SCHEMBL2026104 0.75 BCAT1 (0.55) KEAP1CA1CA2MMP1MMP2
SCHEMBL398043 0.75 TBXA2R (0.42) ALDH1A1CA1CA2MMP1MMP2
SCHEMBL599971 0.75 EPHX2 (0.49) ALDH1A1TSHRMMP1MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113200994-B Application of podophyllotoxin carboxylate derivatives in preparation of anti-tumor products 济宁市第一人民医院 2022-05-17 CN claimed
CN-112010791-B Novel lithospermine phenylacetate derivative containing benzenesulfonamide structural unit and synthesis method and application thereof 济宁市第一人民医院 2022-04-08 CN claimed
CN-113200994-A Application of podophyllotoxin carboxylate derivatives in preparation of anti-tumor products 济宁市第一人民医院 2021-08-03 CN claimed
CN-112010791-A Novel lithospermine phenylacetate derivative containing benzenesulfonamide structural unit and synthesis method and application thereof 济宁市第一人民医院 2020-12-01 CN claimed
CN-113185529-B Preparation method of benzoyl-containing acrylic acid podophyllotoxin ester derivative and application of benzoyl-containing acrylic acid podophyllotoxin ester derivative in tumor inhibition 济宁市第一人民医院 2022-06-21 CN disclosed
CN-113200994-B Application of podophyllotoxin carboxylate derivatives in preparation of anti-tumor products 济宁市第一人民医院 2022-05-17 CN disclosed
CN-113200994-B Application of podophyllotoxin carboxylate derivatives in preparation of anti-tumor products 济宁市第一人民医院 2022-05-17 CN disclosed
CN-113214281-B Synthesis of benzene sulfonamide phenylbutyrate podophyllotoxin ester derivatives and application of benzene sulfonamide phenylbutyrate podophyllotoxin ester derivatives in anticancer drugs 济宁市第一人民医院 2022-05-17 CN disclosed
CN-112010791-B Novel lithospermine phenylacetate derivative containing benzenesulfonamide structural unit and synthesis method and application thereof 济宁市第一人民医院 2022-04-08 CN disclosed
CN-112010791-B Novel lithospermine phenylacetate derivative containing benzenesulfonamide structural unit and synthesis method and application thereof 济宁市第一人民医院 2022-04-08 CN disclosed
CN-113214281-A Synthesis of benzene sulfonamide phenylbutyrate podophyllotoxin ester derivatives and application of benzene sulfonamide phenylbutyrate podophyllotoxin ester derivatives in anticancer drugs 济宁市第一人民医院 2021-08-06 CN disclosed
CN-113200994-A Application of podophyllotoxin carboxylate derivatives in preparation of anti-tumor products 济宁市第一人民医院 2021-08-03 CN disclosed
CN-113200994-A Application of podophyllotoxin carboxylate derivatives in preparation of anti-tumor products 济宁市第一人民医院 2021-08-03 CN disclosed
CN-113185529-A Preparation method of benzoyl-containing acrylic acid podophyllotoxin ester derivative and application of benzoyl-containing acrylic acid podophyllotoxin ester derivative in tumor inhibition 济宁市第一人民医院 2021-07-30 CN disclosed
CN-112010791-A Novel lithospermine phenylacetate derivative containing benzenesulfonamide structural unit and synthesis method and application thereof 济宁市第一人民医院 2020-12-01 CN disclosed
CN-112010791-A Novel lithospermine phenylacetate derivative containing benzenesulfonamide structural unit and synthesis method and application thereof 济宁市第一人民医院 2020-12-01 CN disclosed