SCHEMBL28512436

SCHEMBL28512436

N#Cc1ccnc2c(OS(=O)(=O)C(F)(F)F)cccc12

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.43
PDE4C Q08493 3/20 0.43
PDE4D Q08499 3/20 0.43
SLC22A12 Q96S37 4/20 0.37
AR P10275 1/20 0.37
METAP2 P50579 1/20 0.36
METAP1 P53582 1/20 0.36
DRD2 P14416 4/20 0.34
DRD3 P35462 4/20 0.34
DRD4 P21917 3/20 0.34
SCN9A Q15858 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
DRD1 P21728 2/20 0.33
DRD5 P21918 2/20 0.33
HTR1D P28221 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31156589 0.80 KDM4E (0.43) PDE4APDE4CPDE4DMETAP2METAP1
SCHEMBL24715854 0.75 HTR1A (0.55)
SCHEMBL4443907 0.74 SLC22A12 (0.40) SLC22A12ARDRD2DRD3DRD4
SCHEMBL249779 0.74 METAP2 (0.64) PDE4APDE4CPDE4DMETAP2METAP1
SCHEMBL4818198 0.74 METAP2 (0.42) PDE4APDE4CPDE4DMETAP2METAP1
SCHEMBL1054398 0.74 SLC22A12 (0.37) PDE4APDE4CPDE4DSLC22A12DRD2
SCHEMBL20554633 0.73 SCN9A (0.39) ARSCN9A
SCHEMBL15125330 0.73 DRD2 (0.35) PDE4APDE4CPDE4DMETAP2METAP1
SCHEMBL737308 0.73 SLC40A1 (0.48) PDE4APDE4CPDE4DMETAP2METAP1
SCHEMBL2379509 0.73 SLC40A1 (0.40) PDE4APDE4CPDE4DARL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112300126-A Heterocyclic DNA-PK inhibitors 山东轩竹医药科技有限公司 2021-02-02 CN disclosed