SCHEMBL28515752

SCHEMBL28515752

COC(=O)Oc1c(-c2ccc(Br)cc2)noc1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.51
MAPT P10636 2/20 0.45
TP53 P04637 2/20 0.45
CACNA1F O60840 1/20 0.45
ABCB1 P08183 1/20 0.45
CACNA1D Q01668 1/20 0.45
CACNA1S Q13698 1/20 0.45
CACNA1C Q13936 1/20 0.45
ALDH1A1 P00352 2/20 0.42
HTT P42858 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HKDC1 Q2TB90 1/20 0.41
MCOLN3 Q8TDD5 1/20 0.41
PTGS2 P35354 1/20 0.39
PPARA Q07869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9533937 0.77 ALDH1A1 (0.50) MAPTTP53ALDH1A1HTTSMN1; SMN2
SCHEMBL15951003 0.73 GABRA5 (0.45) RAB9AMAPTCACNA1FABCB1CACNA1D
SCHEMBL9903838 0.72 NPSR1 (0.48) RAB9AMAPTCACNA1FABCB1CACNA1D
SCHEMBL5242546 0.72 KMT2A (0.56) HTTSMN1; SMN2KMT2AMEN1PTGS2
SCHEMBL1246411 0.72 KMT2A (0.56) RAB9AALDH1A1HTTSMN1; SMN2KMT2A
SCHEMBL2470754 0.72 RAB9A (0.54) RAB9AMAPTCACNA1FABCB1CACNA1D
SCHEMBL9533383 0.71 GPBAR1 (0.51) MAPTNPC1KMT2AMEN1POLB
SCHEMBL27495331 0.71 KMT2A (0.55) ALDH1A1HTTSMN1; SMN2KMT2AMEN1
SCHEMBL8594811 0.71 ALDH1A1 (0.35) MAPTALDH1A1HTTSMN1; SMN2KDM4E
SCHEMBL9535701 0.70 KMT2A (0.54) HTTSMN1; SMN2KMT2AMEN1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112041316-B Isoxazole O-linked carbamoyl cyclohexyl acids as LPA antagonists 百时美施贵宝公司 2024-11-22 CN disclosed
CN-112041316-A Isoxazole O-linked carbamoylcyclohexanoic acids as LPA antagonists 百时美施贵宝公司 2020-12-04 CN disclosed