SCHEMBL28518318

SCHEMBL28518318

CCOC(=O)Cn1ccc2ncc(Br)cc21

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
GRIN2B Q13224 19/20 0.47
GRIN1 Q05586 5/20 0.46
CYP2C9 P11712 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22775410 0.78 ALDH1A1 (0.44) KDM4EALDH1A1
SCHEMBL3589940 0.78 GRIN2B (0.51) GRIN2BGRIN1CYP2C9KCNH2
SCHEMBL12291376 0.77 GRIN2B (0.40) GRIN2BGRIN1
SCHEMBL28523558 0.77 GRIN2B (0.77) GRIN2BGRIN1CYP2C9KCNH2
SCHEMBL4485443 0.75 NTSR1 (0.52) ALDH1A1
SCHEMBL18363131 0.74 GRIN2B (0.69) GRIN2B
SCHEMBL18363127 0.74 GRIN2B (0.69) GRIN2B
SCHEMBL20596219 0.74 RAB9A (0.47) KDM4EALDH1A1CYP2C9
SCHEMBL31528647 0.74 FPR2 (0.45) KDM4EALDH1A1CYP2C9
SCHEMBL3046102 0.73 PPARD (0.41) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026094-B Substituted 4-azaindoles and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2021-02-09 CN disclosed