SCHEMBL28520847

SCHEMBL28520847

CC(=O)ON(Cc1ccccc1N)C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 4/20 0.38
FDPS P14324 1/20 0.34
AKT1 P31749 2/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
ITGA4 P13612 1/20 0.32
ITGB7 P26010 1/20 0.32
ATM Q13315 1/20 0.32
ALDH1A1 P00352 2/20 0.32
HSD17B10 Q99714 1/20 0.32
KDM1A O60341 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
RCE1 Q9Y256 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2061803 0.80 SLC6A4 (0.43) FDPSAKT1HDAC3HDAC1HDAC2
SCHEMBL7211228 0.80 FDPS (0.37) L3MBTL1FDPSAKT1HDAC3HDAC1
SCHEMBL27829838 0.78 HDAC3 (0.37) L3MBTL1FDPSAKT1HDAC3HDAC1
SCHEMBL5010708 0.76 AAK1 (0.38) FDPSAKT1HDAC3HDAC1HDAC2
SCHEMBL8605151 0.75 HDAC3 (0.40) L3MBTL1FDPSAKT1HDAC3HDAC1
SCHEMBL5271185 0.74 MTNR1A (0.47) L3MBTL1FDPSALDH1A1HSD17B10KDM4E
SCHEMBL3406057 0.73 HDAC3 (0.39) AKT1HDAC3HDAC1HDAC2NCOR2
SCHEMBL23819882 0.72 RIPK1 (0.47) L3MBTL1HDAC1HDAC2ATMALDH1A1
SCHEMBL2728970 0.72 L3MBTL1 (0.38) L3MBTL1
SCHEMBL6677666 0.71 ESR1 (0.42) L3MBTL1AKT1HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108112251-B NRF2 modulators 葛兰素史克知识产权发展有限公司 2021-03-05 CN disclosed