SCHEMBL28526559

SCHEMBL28526559

COC[C@]1(C=O)CC[C@@H](c2ccccc2)N1C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.40
RIPK1 Q13546 5/20 0.38
GPR119 Q8TDV5 2/20 0.37
NR1H2 P55055 6/20 0.37
NR1H3 Q13133 5/20 0.37
RXRA P19793 2/20 0.37
KDM4E B2RXH2 1/20 0.36
PKM P14618 1/20 0.36
KDM1A O60341 1/20 0.36
RORC P51449 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28518960 0.90 RIPK1 (0.40) ABCB1RIPK1GPR119NR1H2NR1H3
SCHEMBL20835760 0.88 CALCRL (0.38) ABCB1RIPK1KDM1A
SCHEMBL28523788 0.81 ABCB1 (0.46) ABCB1RIPK1GPR119NR1H2NR1H3
SCHEMBL20835514 0.80 ABCB1 (0.40) ABCB1RIPK1GPR119NR1H2NR1H3
SCHEMBL20835558 0.80 ABCB1 (0.38) ABCB1RIPK1GPR119NR1H2NR1H3
SCHEMBL28907234 0.79 PKM (0.41) RIPK1GPR119NR1H2NR1H3RXRA
SCHEMBL16004572 0.78 RORC (0.44) ABCB1RIPK1GPR119NR1H2NR1H3
SCHEMBL28529951 0.78 RIPK1 (0.44) RIPK1GPR119
SCHEMBL20835496 0.78 CALCRL (0.37) ABCB1RIPK1KDM1A
SCHEMBL28285321 0.77 GPR119 (0.43) ABCB1RIPK1GPR119NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109476639-B Pyrrolidine derivatives 橘生药品工业股份有限公司 2021-02-26 CN disclosed