SCHEMBL346337

SCHEMBL346337

CC(C)(C)OC(=O)NC(CCCCNC(=O)c1ccccc1)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.57
TSHR P16473 1/20 0.57
FOLH1 Q04609 12/20 0.53
PPARG P37231 3/20 0.52
PPARA Q07869 3/20 0.52
PPARD Q03181 2/20 0.52
CTSK P43235 3/20 0.52
JAK3 P52333 1/20 0.51
BTK Q06187 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8239220 1.00 ALDH1A1 (0.57) ALDH1A1TSHRFOLH1PPARGPPARA
SCHEMBL2101708 0.96 PPARG (0.59) ALDH1A1TSHRFOLH1PPARGPPARA
SCHEMBL6862461 0.91 NPSR1 (0.54) ALDH1A1TSHRFOLH1
SCHEMBL17550410 0.91 NPSR1 (0.54) ALDH1A1TSHRFOLH1
SCHEMBL16572101 0.89 ALDH1A1 (0.52) ALDH1A1TSHRFOLH1PPARGPPARA
SCHEMBL15625987 0.88 CTSK (0.55) ALDH1A1TSHRPPARGPPARAPPARD
SCHEMBL5970365 0.88 EPHX2 (0.54) ALDH1A1TSHRFOLH1
SCHEMBL2628180 0.86 PPARG (0.53) ALDH1A1TSHRFOLH1PPARGPPARA
SCHEMBL2615858 0.86 PPARG (0.53) ALDH1A1TSHRFOLH1PPARGPPARA
SCHEMBL6865055 0.85 NPSR1 (0.48) ALDH1A1TSHRJAK3BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8338471-B2 (2,5-dioxoimidazolidin-i-yl)-n-hydroxy-acetamides as metalloproteinase inhibitors MEDIVIR AB (SE) 2012-12-25 US disclosed
US-20120015994-A1 (2,5-DIOXOIMIDAZOLIDIN-I-YL)-N-HYDROXY-ACETAMIDES AS METALLOPROTEINASE INHIBITORS MEDIVIR AB (SE) 2012-01-19 US disclosed
US-8022092-B2 (2,5-dioxoimidazolidin-1-yl)-N-hydroxy-acetamides as metalloproteinase inhibitors MEDIVIR AB (SE) 2011-09-20 US disclosed
US-20090215846-A1 (2,5-DIOXOIMIDAZOLIDIN-I-YL)-N-HYDROXY-ACETAMIDES AS METALLOPROTEINASE INHIBITORS MEDIVIR AB (SE) 2009-08-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120015994-A1 (2,5-DIOXOIMIDAZOLIDIN-I-YL)-N-HYDROXY-ACETAMIDES AS METALLOPROTEINASE INHIBITORS MMP12, MMP13, MMP14 ALDH1A1 99/4885TSHR 4332/4885FOLH1 495/4885
US-20090215846-A1 (2,5-DIOXOIMIDAZOLIDIN-I-YL)-N-HYDROXY-ACETAMIDES AS METALLOPROTEINASE INHIBITORS MMP12, MMP13, MMP14 ALDH1A1 99/4885TSHR 4332/4885FOLH1 495/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.