SCHEMBL28533997

SCHEMBL28533997

CCCOC(=O)c1cc(Br)cnc1Cl

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.40
CNR2 P34972 1/20 0.39
OPRK1 P41145 1/20 0.39
THRB P10828 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
ATM Q13315 1/20 0.39
MAPT P10636 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
GABRA2 P47869 1/20 0.38
GABRB2 P47870 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21596476 0.89 OPRK1 (0.40) ALDH1A1KDM4EOPRK1TP53RXFP1
SCHEMBL2782609 0.88 OPRK1 (0.48) ALDH1A1KDM4EOPRK1SMN1; SMN2HSD17B10
SCHEMBL21596477 0.85 OPRK1 (0.40) KDM4EOPRK1THRBMAPTTP53
SCHEMBL20472461 0.82 ALDH1A1 (0.50) ALDH1A1KDM4ECNR2OPRK1ATM
SCHEMBL28522607 0.82 ALDH1A1 (0.46) ALDH1A1KDM4EMAPTLMNATP53
SCHEMBL733159 0.80 OPRK1 (0.49) OPRK1
SCHEMBL17845871 0.78 CYP3A4 (0.47) ALDH1A1KDM4EOPRK1RXFP1SMN1; SMN2
SCHEMBL27734476 0.76 HSP90AB1 (0.36) ALDH1A1KDM4ECNR2OPRK1HTT
SCHEMBL28526753 0.76 ATR (0.38) ALDH1A1OPRK1GABRA2GABRB2
SCHEMBL16077093 0.76 OPRK1 (0.40) OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112334457-A Process for preparing tricyclic compounds 拜耳公司 2021-02-05 CN disclosed