SCHEMBL28537323

SCHEMBL28537323

NC(=O)c1cc2c(ccc3ccccc32)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 3/20 0.48
DYRK1A Q13627 3/20 0.48
CHEK1 O14757 2/20 0.48
AURKA O14965 2/20 0.48
DAPK3 O43293 2/20 0.48
PIM1 P11309 2/20 0.48
FGFR1 P11362 2/20 0.48
PRKACA P17612 2/20 0.48
FLT1 P17948 2/20 0.48
KDR P35968 2/20 0.48
MAPK8 P45983 2/20 0.48
GSK3A P49840 2/20 0.48
GSK3B P49841 2/20 0.48
RPS6KA3 P51812 2/20 0.48
CDK5 Q00535 2/20 0.48
PRKAA1 Q13131 2/20 0.48
ROCK1 Q13464 2/20 0.48
AURKB Q96GD4 2/20 0.48
PLK4 O00444 1/20 0.48
CHEK2 O96017 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9567942 0.85 F9 (0.57) PLAUF9F10
Hydrochloric Acid SCHEMBL9432197 0.83 PLAU (0.58) PLAUF9F10
SCHEMBL9431295 0.80 ALDH1A1 (0.60) DYRK1AGSK3AGSK3BAURKBRPS6KB1
SCHEMBL28540745 0.78 KDM4E (0.61) LIMK1DYRK1ACHEK1AURKADAPK3
SCHEMBL347544 0.77 BCL2L1 (0.69) LIMK1DYRK1ACHEK1AURKADAPK3
SCHEMBL29366392 0.77 BCL2L1 (0.69) LIMK1DYRK1ACHEK1AURKADAPK3
SCHEMBL28744296 0.76 KDM4E (0.59) MAPK1CNR2F9KDM4EGLA
Hydrochloric Acid SCHEMBL2196804 0.75 BCL2L1 (0.67) LIMK1DYRK1ACHEK1AURKADAPK3
SCHEMBL28162040 0.74 DYRK1A (0.51) LIMK1DYRK1ACHEK1AURKADAPK3
SCHEMBL17934651 0.73 ALDH1A1 (0.48) MAPTHPGDTSHRHSD17B10TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108727416-B Tricyclic heteroaromatic amide derivative and preparation and application thereof 北京大学 2021-03-09 CN disclosed