SCHEMBL28540474

SCHEMBL28540474

Fc1cc(F)c(Br)c(CBr)c1

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.39
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13068931 0.79 GPR84 (0.38) GPR84CES2CES1
SCHEMBL28816037 0.79 GPR84 (0.38) GPR84
SCHEMBL29629074 0.79 GPR84 (0.38) GPR84CES2CES1
SCHEMBL489929 0.78 RIPK1 (0.41) GPR84CES2CES1
SCHEMBL919665 0.76 KDM1A (0.42) GPR84CES2CES1
SCHEMBL33526163 0.76 GPR84 (0.36) GPR84
SCHEMBL5162621 0.74 RAPGEF4 (0.32) GPR84
SCHEMBL20594895 0.74 GPR84 (0.31) GPR84
SCHEMBL6553272 0.73 KDM1A (0.41) GPR84CES2CES1
SCHEMBL24357673 0.72 KDM1A (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108349983-B Dihydroimidazopyrazinone derivatives useful for the treatment of cancer 阿斯利康(瑞典)有限公司 2021-02-26 CN disclosed
CN-108349983-A The useful glyoxalidine for the treatment of cancer and pyrazinone derivatives 阿斯利康(瑞典)有限公司 2018-07-31 CN disclosed