SCHEMBL2854501

SCHEMBL2854501

O=C(Nc1nc2ccccc2[nH]1)Oc1cnn(-c2ccccn2)c1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.43
LMNA P02545 2/20 0.41
CYP3A4 P08684 1/20 0.41
NPC1 O15118 9/20 0.40
RAB9A P51151 8/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
TP53 P04637 3/20 0.40
ALDH1A1 P00352 1/20 0.40
ALOX12 P18054 1/20 0.40
PKM P14618 4/20 0.39
HSP90AA1 P07900 1/20 0.39
PAX8 Q06710 1/20 0.39
MAOB P27338 1/20 0.39
ADORA2A P29274 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
GAA P10253 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853272 0.89 MTOR (0.48) MTORLMNACYP3A4NPC1RAB9A
SCHEMBL2858021 0.88 MTOR (0.42) MTORLMNACYP3A4NPC1RAB9A
SCHEMBL2858176 0.85 MTOR (0.42) MTORLMNACYP3A4NPC1RAB9A
SCHEMBL2857349 0.83 ABCB1 (0.49) MTORLMNACYP3A4NPC1RAB9A
SCHEMBL2854611 0.79 TRPV1 (0.41) LMNANPC1RAB9ASMN1; SMN2TP53
SCHEMBL2856635 0.77 MALT1 (0.42) ALDH1A1KDM4E
SCHEMBL2857586 0.77 ATR (0.39) NPC1RAB9ASMN1; SMN2TP53ALDH1A1
SCHEMBL2854810 0.76 KMT2A (0.46) MTORLMNANPC1RAB9AALDH1A1
SCHEMBL2855796 0.76 ALDH1A1 (0.43) LMNANPC1RAB9ASMN1; SMN2TP53
SCHEMBL2862979 0.76 TRPV1 (0.44) SMN1; SMN2GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed