SCHEMBL28545324

SCHEMBL28545324

O=C(O)c1ccc(COCCCCl)c([N+](=O)[O-])c1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.50
TSHR P16473 2/20 0.47
LMNA P02545 1/20 0.47
HCAR3 P49019 10/20 0.45
PLA2G4B P0C869 1/20 0.44
APEX1 P27695 1/20 0.44
PDK1 Q15118 1/20 0.44
PRSS1 P07477 1/20 0.43
ALOX5 P09917 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16129649 0.86 HCAR3 (0.56) CASP6TSHRLMNAHCAR3
SCHEMBL16129686 0.85 CASP6 (0.54) CASP6TSHRLMNAHCAR3APEX1
SCHEMBL177446 0.84 HCAR3 (0.53) CASP6TSHRLMNAHCAR3PLA2G4B
SCHEMBL17511817 0.83 HCAR3 (0.58) CASP6TSHRLMNAHCAR3
SCHEMBL28543354 0.81 PRSS1 (0.64) CASP6TSHRLMNAHCAR3PLA2G4B
SCHEMBL28748754 0.81 HCAR3 (0.51) CASP6TSHRLMNAHCAR3PDK1
SCHEMBL2292095 0.79 CASP6 (0.64) CASP6TSHRLMNAHCAR3APEX1
SCHEMBL4175596 0.78 CASP6 (0.58) CASP6TSHRLMNAHCAR3APEX1
SCHEMBL6476753 0.78 TSHR (0.51) CASP6TSHRLMNAHCAR3PLA2G4B
SCHEMBL23978245 0.77 MAOB (0.60) CASP6TSHRLMNAHCAR3ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109503518-B Substituted biaryl amide compound and preparation method and application thereof 中国医学科学院医药生物技术研究所 2021-03-30 CN disclosed
CN-109503518-A A kind of substituted double aromatic radical amide compounds and its preparation method and application 中国医学科学院医药生物技术研究所 2019-03-22 CN disclosed