SCHEMBL28548823

SCHEMBL28548823

C[C@H](c1ccnc(C(N)=O)c1)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.38
OPRM1 P35372 4/20 0.37
SCN10A Q9Y5Y9 3/20 0.37
NR3C2 P08235 1/20 0.36
DEGS1 O15121 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
TSHR P16473 1/20 0.36
MC4R P32245 1/20 0.36
ADRA1A P35348 1/20 0.36
MC3R P41968 1/20 0.36
GSK3B P49841 1/20 0.36
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
RAF1 P04049 1/20 0.35
IGF1R P08069 1/20 0.35
GRM2 Q14416 2/20 0.35
LOXL2 Q9Y4K0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13847046 0.84 DEGS1 (0.32) DEGS1
SCHEMBL13028405 0.82 NPSR1 (0.32) DEGS1
SCHEMBL2332478 0.82 NPSR1 (0.32) DEGS1
SCHEMBL25687807 0.82 ADORA3 (0.41) KMT2AOPRM1NR3C2ADORA3TSHR
SCHEMBL10204249 0.82 RAF1 (0.43) OPRM1NR3C2ADORA3TSHRMC4R
SCHEMBL3439404 0.76 ALDH1A1 (0.42) KMT2AOPRM1NR3C2ADORA3TSHR
SCHEMBL22888217 0.76 KMT2A (0.54) KMT2ADEGS1ADORA3TSHRMC4R
SCHEMBL2324988 0.75 OPRM1 (0.37) OPRM1NR3C2ADORA3TSHRMC4R
SCHEMBL568385 0.73 OPRM1 (0.38) OPRM1NR3C2ADORA3TSHRMC4R
SCHEMBL17411826 0.73 GABRP (0.36) DEGS1TSHRGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112638896-A ASK1 inhibitors 比奥根MA公司 2021-04-09 CN disclosed