SCHEMBL2855591

SCHEMBL2855591

O=C(NCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Oc1cnn(-c2ccc(Cl)nn2)c1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.41
JUN P05412 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
P2RX1 P51575 1/20 0.39
TMPRSS4 Q9NRS4 1/20 0.39
TACR1 P25103 3/20 0.38
CCR1 P32246 5/20 0.37
MTOR P42345 1/20 0.37
MLYCD O95822 1/20 0.36
HPGD P15428 2/20 0.35
P2RX7 Q99572 1/20 0.35
ALDH1A1 P00352 3/20 0.35
GAA P10253 2/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2857181 0.92 CCR1 (0.47) CCR1HPGDGAALMNACYP1A2
SCHEMBL2854487 0.88 TSHR (0.45) CCR1HPGDP2RX7ALDH1A1LMNA
SCHEMBL2859076 0.84 KEAP1 (0.42) CCR1ALDH1A1
SCHEMBL2856252 0.84 P2RX1 (0.49) CCR2JUNNFKB1NFKB2RELA
SCHEMBL2853270 0.84 CCR1 (0.51) P2RX1TMPRSS4TACR1CCR1P2RX7
SCHEMBL2857977 0.83 ALDH1A1 (0.47) HPGDALDH1A1KDM4ELMNAPOLB
SCHEMBL2857994 0.83 MTOR (0.46) TACR1CCR1MTORMLYCDP2RX7
SCHEMBL2857073 0.82 CCR1 (0.48) CCR2TACR1CCR1ALDH1A1KDM4E
SCHEMBL2855603 0.82 P2RX1 (0.44) P2RX1TMPRSS4TACR1CCR1MTOR
SCHEMBL2857615 0.82 MTOR (0.37) MTORP2RX7LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed