SCHEMBL2856282

SCHEMBL2856282

COc1ccc(CNC(=O)c2cnn(-c3ccccn3)c2C(F)(F)F)c(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT2 Q96PD7 2/20 0.54
TAS1R3 Q7RTX0 2/20 0.51
TAS1R1 Q7RTX1 2/20 0.51
PDE4B Q07343 1/20 0.51
EPHX2 P34913 2/20 0.49
KLKB1 P03952 1/20 0.49
ALDH1A1 P00352 3/20 0.49
HPGD P15428 2/20 0.49
GAA P10253 1/20 0.49
PKM P14618 1/20 0.49
HTT P42858 1/20 0.49
NPSR1 Q6W5P4 2/20 0.48
TSHR P16473 1/20 0.48
MAPK8 P45983 1/20 0.46
MALT1 Q9UDY8 1/20 0.44
MAPT P10636 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
THRB P10828 1/20 0.44
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850370 0.90 DGAT2 (0.55) DGAT2TAS1R3TAS1R1PDE4BEPHX2
SCHEMBL2859103 0.87 EPHX2 (0.45) DGAT2TAS1R3TAS1R1PDE4BEPHX2
SCHEMBL2852021 0.86 DGAT2 (0.51) DGAT2TAS1R3TAS1R1PDE4BEPHX2
SCHEMBL2850896 0.83 DGAT2 (0.57) DGAT2TAS1R3TAS1R1PDE4BEPHX2
SCHEMBL2856352 0.82 DGAT2 (0.56) DGAT2TAS1R3TAS1R1PDE4BEPHX2
SCHEMBL10364566 0.78 KDM4E (0.52) ALDH1A1HPGDMALT1MAPTKMT2A
SCHEMBL2857544 0.77 TSHR (0.45) DGAT2TAS1R3TAS1R1PDE4BEPHX2
SCHEMBL2855742 0.76 CCR1 (0.58) HPGDGAAMEN1KMT2A
SCHEMBL2857426 0.75 CCR1 (0.55) DGAT2ALDH1A1HPGDHTTNPSR1
SCHEMBL2852937 0.74 KLKB1 (0.43) DGAT2TAS1R3TAS1R1PDE4BEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed