SCHEMBL2857544

SCHEMBL2857544

COc1ccc(CNC(=O)Oc2cnn(-c3ncccn3)c2C(F)(F)F)c(OC)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.45
ALDH1A1 P00352 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TAS1R3 Q7RTX0 2/20 0.44
TAS1R1 Q7RTX1 2/20 0.44
PDE4B Q07343 1/20 0.44
KLKB1 P03952 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MAPK1 P28482 1/20 0.42
DGAT2 Q96PD7 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
ALOX15 P16050 2/20 0.40
CYP2C19 P33261 2/20 0.40
USP2 O75604 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
KDM4C Q9H3R0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2859103 0.90 EPHX2 (0.45) TSHRALDH1A1NPSR1TAS1R3TAS1R1
SCHEMBL2850370 0.86 DGAT2 (0.55) TSHRALDH1A1NPSR1TAS1R3TAS1R1
SCHEMBL2853809 0.85 P2RX7 (0.49) TSHRALDH1A1NPSR1TAS1R3TAS1R1
SCHEMBL2853175 0.85 KLKB1 (0.43) TSHRALDH1A1NPSR1TAS1R3TAS1R1
SCHEMBL2852937 0.84 KLKB1 (0.43) TSHRALDH1A1NPSR1TAS1R3TAS1R1
SCHEMBL2855496 0.79 KDM4E (0.46) TSHRALDH1A1NPSR1KDM4EMAPK1
SCHEMBL2855714 0.77 EPHX1 (0.45) NPSR1MAPK1MEN1KMT2AMAPT
SCHEMBL2856282 0.77 DGAT2 (0.54) TSHRALDH1A1NPSR1TAS1R3TAS1R1
SCHEMBL2850129 0.76 ALDH1A1 (0.52) ALDH1A1KDM4EMAPK1KMT2ACYP1A2
SCHEMBL2852117 0.76 P2RX7 (0.48) ALDH1A1MEN1KMT2AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed