SCHEMBL28564709

SCHEMBL28564709

NC(=O)Cc1csc2ccc(F)cc12

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.57
MTNR1B P49286 1/20 0.57
CA2 P00918 1/20 0.56
KEAP1 Q14145 1/20 0.50
NFE2L2 Q16236 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.47
ICMT O60725 3/20 0.44
CYP2A6 P11509 2/20 0.41
MPO P05164 3/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 2/20 0.40
SLC6A4 P31645 1/20 0.40
JUN P05412 1/20 0.39
MAPK8 P45983 1/20 0.39
MAPK9 P45984 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31164712 1.00 MTNR1A (0.57) MTNR1AMTNR1BCA2KEAP1NFE2L2
SCHEMBL22499949 0.86 KEAP1 (0.68) MTNR1AMTNR1BCA2KEAP1NFE2L2
SCHEMBL9751552 0.81 CA2 (0.56) MTNR1AMTNR1BCA2KEAP1NFE2L2
SCHEMBL6202916 0.81 KEAP1 (0.75) CA2KEAP1NFE2L2SMN1; SMN2CYP2A6
SCHEMBL28563290 0.81 CYP2A6 (0.64) MTNR1AMTNR1BCA2KEAP1NFE2L2
SCHEMBL8605628 0.79 MTNR1A (0.59) MTNR1AMTNR1BCA2KEAP1NFE2L2
SCHEMBL31164737 0.79 MTNR1A (0.54) MTNR1AMTNR1BCA2KEAP1NFE2L2
SCHEMBL10982992 0.79 MTNR1A (0.54) MTNR1AMTNR1BCA2KEAP1NFE2L2
SCHEMBL4605763 0.78 CYP2A6 (0.64) MTNR1AMTNR1BCA2KEAP1NFE2L2
SCHEMBL6003503 0.78 MTNR1A (0.60) MTNR1AMTNR1BCA2KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025122501-A1 BENZOTHIOPHENE-3-YL- AND BENZOSELENOPHENE-3-YL (BICLYCLIC HETEROARYL) MALEMIDES AS GSK-3 INHIBITORS MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2025-06-12 WO disclosed
CN-108264509-B Substituted benzothieno [2,3-c ] tetrahydropyridine derivatives, preparation method and application thereof 复旦大学 2021-05-04 CN disclosed