SCHEMBL28563290

SCHEMBL28563290

NC(=O)Cc1csc2ccc(Br)cc12

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.64
CA2 P00918 2/20 0.56
HDAC10 Q969S8 1/20 0.52
HDAC11 Q96DB2 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
KEAP1 Q14145 1/20 0.50
NFE2L2 Q16236 1/20 0.50
MAPT P10636 3/20 0.47
UTS2R Q9UKP6 1/20 0.43
LMNA P02545 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
TP53 P04637 1/20 0.39
JUN P05412 1/20 0.39
MAPK8 P45983 1/20 0.39
MAPK9 P45984 1/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
EPHX1 P07099 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7429693 0.86 KEAP1 (0.68) CYP2A6CA2HDAC10HDAC11HDAC8
SCHEMBL9751552 0.81 CA2 (0.56) CYP2A6CA2KEAP1NFE2L2MAPT
SCHEMBL31164712 0.81 MTNR1A (0.57) CYP2A6CA2KEAP1NFE2L2MAPT
SCHEMBL28564709 0.81 MTNR1A (0.57) CYP2A6CA2KEAP1NFE2L2MAPT
SCHEMBL6202916 0.81 KEAP1 (0.75) CYP2A6CA2KEAP1NFE2L2MAPT
SCHEMBL15897090 0.81 CYP2A6 (0.55) CYP2A6CA2HDAC10HDAC11HDAC8
SCHEMBL30469746 0.81 CYP2A6 (0.55) CYP2A6CA2HDAC10HDAC11HDAC8
SCHEMBL8605628 0.79 MTNR1A (0.59) CYP2A6CA2KEAP1NFE2L2LMNA
SCHEMBL28566065 0.79 CYP2A6 (0.52) CYP2A6CA2HDAC10HDAC11HDAC8
SCHEMBL31425881 0.79 CYP2A6 (0.52) CYP2A6CA2HDAC10HDAC11HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108264509-B Substituted benzothieno [2,3-c ] tetrahydropyridine derivatives, preparation method and application thereof 复旦大学 2021-05-04 CN disclosed