SCHEMBL28593231

SCHEMBL28593231

COC(=O)c1nc(-c2cccnc2)sc1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.52
CYP3A4 P08684 3/20 0.52
CYP2C19 P33261 2/20 0.52
LMNA P02545 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.49
CYP19A1 P11511 1/20 0.48
CYP11B1 P15538 1/20 0.48
CYP11B2 P19099 1/20 0.48
KDM4E B2RXH2 4/20 0.48
ALDH1A1 P00352 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
HPGD P15428 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CDC7 O00311 2/20 0.47
DBF4 Q9UBU7 2/20 0.47
CFTR P13569 1/20 0.46
MAPT P10636 1/20 0.46
CISD2 Q8N5K1 1/20 0.45
MEN1 O00255 1/20 0.44
CYP2D6 P10635 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL289392 0.86 CDC7 (0.60) CYP1A2CYP3A4CYP2C19LMNAKDM4E
SCHEMBL15109222 0.85 CYP3A4 (0.56) CYP1A2CYP3A4CYP2C19LMNACYP19A1
SCHEMBL28801535 0.85 L3MBTL1 (0.66) LMNAL3MBTL1KDM4EALDH1A1SMN1; SMN2
SCHEMBL14059574 0.83 CYP3A4 (0.60) CYP1A2CYP3A4CYP2C19LMNACYP19A1
SCHEMBL18055899 0.78 L3MBTL1 (0.48) CYP1A2L3MBTL1KDM4EALDH1A1SMN1; SMN2
SCHEMBL14237794 0.76 CYP1A2 (0.57) CYP1A2CYP3A4CYP2C19LMNACYP19A1
SCHEMBL2484432 0.76 ATR (0.67) CYP3A4
SCHEMBL11388698 0.75 ALDH1A1 (0.51) CYP1A2CYP3A4CYP2C19LMNACYP19A1
SCHEMBL17629283 0.75 PAX8 (0.43) CYP1A2CYP3A4CYP2C19LMNAL3MBTL1
SCHEMBL18569364 0.74 CDC7 (0.58) CYP1A2CYP3A4CYP2C19LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107001349-B Herbicidal pyrido/pyrimidothiazoles 先正达参股股份有限公司 2021-07-02 CN disclosed