SCHEMBL28596272

SCHEMBL28596272

CN1C(=O)C(=[N+]=[N-])c2cccc(F)c21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 2/20 0.40
POLB P06746 1/20 0.40
CHRM5 P08912 2/20 0.35
TRPA1 O75762 1/20 0.34
CHRM1 P11229 2/20 0.33
CASP3 P42574 1/20 0.33
BRD4 O60885 1/20 0.33
USP2 O75604 2/20 0.33
CASP1 P29466 1/20 0.33
BRCA1 P38398 1/20 0.33
CASP7 P55210 1/20 0.33
TTR P02766 1/20 0.33
CES1 P23141 1/20 0.33
PKM P14618 1/20 0.32
ATM Q13315 1/20 0.31
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20534377 0.81 ALDH1A1 (0.40) MEN1KMT2AALDH1A1POLBCASP3
SCHEMBL28593612 0.81 ALDH1A1 (0.41) MEN1KMT2AALDH1A1POLBCHRM5
SCHEMBL29785238 0.78 ALDH1A1 (0.65) MEN1KMT2AALDH1A1POLBCHRM5
SCHEMBL2816698 0.78 ALDH1A1 (0.65) MEN1KMT2AALDH1A1POLBCHRM5
SCHEMBL28428472 0.77 HSPA1A (0.39) MEN1KMT2AALDH1A1POLBCHRM5
SCHEMBL11265954 0.73 TTR (0.58) MEN1KMT2AALDH1A1TRPA1CASP3
SCHEMBL20534453 0.68 PARK7 (0.36) MEN1KMT2AALDH1A1CASP3BRD4
SCHEMBL20534614 0.68 CA1 (0.44) CHRM5TRPA1CASP3BRD4CASP1
SCHEMBL5001267 0.67 CHRM5 (0.60) MEN1KMT2AALDH1A1POLBCHRM5
SCHEMBL5502497 0.66 MEN1 (0.49) MEN1KMT2AALDH1A1POLBCHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111961060-B Preparation method of spiroheterocyclic 2, 3-dihydrobenzofuran compound with optical activity 遵义医科大学 2021-07-06 CN disclosed
CN-111961060-A Preparation method of spiroheterocyclic 2, 3-dihydrobenzofuran compound with optical activity 遵义医科大学 2020-11-20 CN disclosed