SCHEMBL28601296

SCHEMBL28601296

CC(NC(=O)c1ccc(-c2ccccc2)nc1)c1ccccc1Cl

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BAZ2B Q9UIF8 1/20 0.58
ROCK2 O75116 7/20 0.51
ROCK1 Q13464 3/20 0.51
HPGDS O60760 2/20 0.50
MAPK3 P27361 1/20 0.50
MAPK1 P28482 1/20 0.50
LDHA P00338 1/20 0.50
PRKG1 Q13976 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
CTSA P10619 3/20 0.47
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16496342 0.83 BAZ2B (0.65) BAZ2BROCK2ROCK1HPGDSMAPK1
SCHEMBL28601974 0.83 MEN1 (0.61) ROCK2ROCK1HPGDSMAPK3MAPK1
SCHEMBL16495348 0.79 CTSA (0.56) BAZ2BMEN1KMT2ACTSA
SCHEMBL28598671 0.79 CTSA (0.59) ROCK2ROCK1MAPK3MAPK1CYP1A2
SCHEMBL28603586 0.77 KMO (0.51) ROCK2ROCK1MAPK3MAPK1CTSA
SCHEMBL16496169 0.76 BAZ2B (0.62) BAZ2BROCK2HPGDSLDHAPRKG1
SCHEMBL16496172 0.76 BAZ2B (0.62) BAZ2BROCK2HPGDSLDHAPRKG1
SCHEMBL16495423 0.76 NPC1 (0.69) BAZ2BROCK2ROCK1HPGDSMAPK1
SCHEMBL16495693 0.75 ROCK2 (0.60) BAZ2BROCK2ROCK1HPGDSMAPK1
SCHEMBL28611023 0.75 TUBB4A (0.50) ROCK2ROCK1MAPK3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110407824-B Aryl formamide compound and preparation method, pharmaceutical composition and application thereof 安徽医科大学 2021-07-02 CN disclosed