SCHEMBL28617460

SCHEMBL28617460

C=CC(=O)Nc1ccc(C(=O)N[C@H](c2ccccc2)C(C)C)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.63
TGM2 P21980 5/20 0.53
ALDH1A1 P00352 4/20 0.51
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
HDAC3 O15379 3/20 0.48
HDAC4 P56524 3/20 0.48
HDAC7 Q8WUI4 3/20 0.48
HDAC2 Q92769 3/20 0.48
HDAC10 Q969S8 3/20 0.48
HDAC11 Q96DB2 3/20 0.48
HDAC8 Q9BY41 3/20 0.48
HDAC6 Q9UBN7 3/20 0.48
HDAC9 Q9UKV0 3/20 0.48
HDAC5 Q9UQL6 3/20 0.48
LMNA P02545 3/20 0.48
TP53 P04637 1/20 0.48
HPGD P15428 1/20 0.47
POLB P06746 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28617369 0.87 KMT2A (0.60) TGM2ALDH1A1MEN1KMT2ALMNA
SCHEMBL28619644 0.87 KMT2A (0.60) TGM2ALDH1A1MEN1KMT2ALMNA
SCHEMBL28630813 0.87 KMT2A (0.60) TGM2ALDH1A1MEN1KMT2ALMNA
SCHEMBL28630765 0.79 RAB9A (0.62) TGM2ALDH1A1MEN1KMT2ALMNA
SCHEMBL28620836 0.76 MAPK1 (0.48) ALDH1A1MEN1KMT2ALMNANPC1
SCHEMBL28616230 0.76 NPC1 (0.52) TGM2ALDH1A1MEN1KMT2ALMNA
SCHEMBL21179425 0.75 TGM2 (0.50) TGM2MEN1KMT2ALMNANPC1
SCHEMBL28615912 0.74 TGM2 (0.61) TGM2ALDH1A1MEN1KMT2ALMNA
SCHEMBL28620280 0.74 TGM2 (0.61) TGM2ALDH1A1MEN1KMT2ALMNA
SCHEMBL17327878 0.74 TGM2 (0.63) TGM2MEN1KMT2ALMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109438279-B Small molecule compound for overcoming EGFR drug-resistant mutation and preparation method and application thereof 四川大学 2021-08-31 CN disclosed