SCHEMBL28630765

SCHEMBL28630765

C=CC(=O)Nc1ccc(C(=O)N[C@@H](C)Cc2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.62
NPC1 O15118 3/20 0.62
SMN1; SMN2 Q16637 3/20 0.57
KMT2A Q03164 3/20 0.57
MEN1 O00255 2/20 0.57
TP53 P04637 1/20 0.57
HTT P42858 1/20 0.52
TGM2 P21980 3/20 0.51
TAAR1 Q96RJ0 1/20 0.51
HPGD P15428 1/20 0.49
KDM4E B2RXH2 1/20 0.48
MAPT P10636 1/20 0.48
HSP90AA1 P07900 1/20 0.47
POLB P06746 1/20 0.47
ACACB O00763 2/20 0.46
LMNA P02545 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9694817 0.81 TAAR1 (0.69) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL11949543 0.81 RAB9A (0.79) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL880676 0.81 RAB9A (0.79) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL28630813 0.81 KMT2A (0.60) NPC1SMN1; SMN2KMT2AMEN1TP53
SCHEMBL28617369 0.81 KMT2A (0.60) NPC1SMN1; SMN2KMT2AMEN1TP53
SCHEMBL28619644 0.81 KMT2A (0.60) NPC1SMN1; SMN2KMT2AMEN1TP53
SCHEMBL4103656 0.80 RAB9A (0.74) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL28617460 0.79 HDAC1 (0.63) NPC1KMT2AMEN1TP53TGM2
SCHEMBL28616232 0.78 HDAC6 (0.59) RAB9ATP53TGM2HPGDKDM4E
SCHEMBL23099741 0.77 NPC1 (0.74) RAB9ANPC1SMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109438279-B Small molecule compound for overcoming EGFR drug-resistant mutation and preparation method and application thereof 四川大学 2021-08-31 CN disclosed