SCHEMBL28623786

SCHEMBL28623786

COc1nc(-c2cccnc2)ccc1C=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.52
ERN1 O75460 3/20 0.51
RAB9A P51151 3/20 0.49
ALDH1A1 P00352 2/20 0.49
HSD17B10 Q99714 2/20 0.49
GAA P10253 1/20 0.49
TSHR P16473 1/20 0.49
CYP2A6 P11509 3/20 0.46
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.46
SQOR Q9Y6N5 1/20 0.46
CYP3A4 P08684 2/20 0.44
CYP2E1 P05181 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2B6 P20813 1/20 0.44
CYP2C19 P33261 1/20 0.44
CYP19A1 P11511 3/20 0.43
ATM Q13315 1/20 0.42
CYP17A1 P05093 2/20 0.42
CYP11B2 P19099 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4799732 0.84 SQOR (0.49) NPC1RAB9AALDH1A1HSD17B10GAA
SCHEMBL30772447 0.84 SQOR (0.49) NPC1RAB9AALDH1A1HSD17B10GAA
SCHEMBL12427715 0.82 SQOR (0.46) NPC1RAB9AALDH1A1HSD17B10GAA
SCHEMBL5782678 0.77 ERN1 (0.61) NPC1ERN1RAB9AALDH1A1CYP2A6
SCHEMBL28362190 0.75 ERN1 (0.47) NPC1ERN1ALDH1A1CYP2A6CYP3A4
SCHEMBL12427721 0.74 KDM1A (0.45) ALDH1A1HSD17B10GAAKDM4EHPGD
SCHEMBL19737563 0.73 TTK (0.49) NPC1ERN1ALDH1A1CYP2A6CYP3A4
SCHEMBL7677974 0.73 ERN1 (0.69) NPC1ERN1RAB9AALDH1A1HSD17B10
SCHEMBL19737559 0.72 LIMK1 (0.48) NPC1ERN1RAB9ACYP2A6KDM4E
SCHEMBL12427716 0.72 F2RL3 (0.40) RAB9AALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117327078-A Heterocyclic compound, pharmaceutical composition containing same, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2024-01-02 CN disclosed
CN-117263945-A Heterocyclic compound, pharmaceutical composition containing same, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-12-22 CN disclosed
CN-113316578-B Heterocyclic compound, pharmaceutical composition containing same, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-10-31 CN disclosed
CN-113316578-A Heterocyclic compounds, pharmaceutical compositions containing them, processes for their preparation and their use 四川科伦博泰生物医药股份有限公司 2021-08-27 CN disclosed