SCHEMBL28627930

SCHEMBL28627930

COC(=O)c1ccc(N)cc1C(=O)OC(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.58
KDM4E B2RXH2 7/20 0.46
ALDH1A1 P00352 5/20 0.46
HSD17B10 Q99714 3/20 0.46
MAPT P10636 3/20 0.46
GLA P06280 3/20 0.46
HPGD P15428 2/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
ATM Q13315 1/20 0.46
CFTR P13569 2/20 0.45
ABL1 P00519 1/20 0.45
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA9 Q16790 3/20 0.41
CA12 O43570 2/20 0.41
CA7 P43166 2/20 0.41
CA14 Q9ULX7 2/20 0.41
PDK2 Q15119 1/20 0.41
PDK4 Q16654 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1403643 0.88 GAA (0.72) GAAKDM4EALDH1A1HSD17B10MAPT
SCHEMBL7623605 0.86 GAA (0.70) GAAKDM4EALDH1A1HSD17B10MAPT
SCHEMBL436207 0.85 ALDH1A1 (0.51) GAAKDM4EALDH1A1HSD17B10MAPT
Dimethyl Phthalate SCHEMBL28028655 0.83 GAA (0.66) GAAKDM4EALDH1A1HSD17B10MAPT
SCHEMBL27622981 0.83 KDM4E (0.47) GAAKDM4EALDH1A1HSD17B10MAPT
SCHEMBL2874165 0.82 KDM4E (0.56) GAAKDM4EALDH1A1HSD17B10MAPT
SCHEMBL1185611 0.81 KMT2A (0.52) GAAKDM4EALDH1A1HSD17B10MAPT
SCHEMBL29439802 0.81 KDM4E (0.47) GAAKDM4EALDH1A1HSD17B10MAPT
SCHEMBL1100205 0.81 ALDH1A1 (0.63) GAAKDM4EALDH1A1MAPTTSHR
SCHEMBL6177925 0.80 CASP1 (0.41) GAAKDM4EALDH1A1HSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113350296-B PAD4 inhibitor loaded by CRGD sequence peptide modified chitosan and preparation method and application thereof 首都医科大学 2022-07-15 CN disclosed
CN-113350296-A PAD4 inhibitor loaded by CRGD sequence peptide modified chitosan and preparation method and application thereof 首都医科大学 2021-09-07 CN disclosed