Chelerythrine

Chelerythrine

SCHEMBL28629157

COc1ccc2c(c[n+](C)c3c4cc5c(cc4ccc23)OCO5)c1OC.C[n+]1cc2c3c(ccc2c2ccc4cc5c(cc4c21)OCO5)OCO3.[Cl-].[Cl-]

nearest known ligand 0.88

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEBDKRB2CHRM1CHRM2CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNGGUCY1A1GUCY1A2GUCY1B1GUCY1B2NAMPTPTAFRSLC10A2SLC6A2SLC6A3TACR1dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Chelerythrine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 5/20 0.88
CHRM1 known ✓ P11229 2/20 0.46
ALDH1A1 P00352 8/20 0.88
MAPT P10636 8/20 0.88
SMN1; SMN2 Q16637 8/20 0.88
HPGD P15428 6/20 0.88
KMT2A Q03164 6/20 0.88
LMNA P02545 6/20 0.88
BAD Q92934 6/20 0.88
MAPK1 P28482 5/20 0.88
BCHE P06276 5/20 0.88
RAC1 P63000 4/20 0.88
POLB P06746 3/20 0.88
NPSR1 Q6W5P4 3/20 0.88
GMNN O75496 2/20 0.88
BLM P54132 2/20 0.88
PMP22 Q01453 2/20 0.88
PRKCE Q02156 1/20 0.88
MEN1 O00255 5/20 0.86
CYP3A4 P08684 5/20 0.86

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chelerythrine SCHEMBL30207103 0.94 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2HPGDKMT2A
Chelerythrine SCHEMBL195109 0.94 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2HPGDKMT2A
Chelerythrine SCHEMBL30527167 0.93 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2HPGDKMT2A
Chelerythrine SCHEMBL288915 0.93 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2HPGDKMT2A
Chelerythrine SCHEMBL30527168 0.93 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2HPGDKMT2A
Chelerythrine SCHEMBL29357531 0.93 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2HPGDKMT2A
Chelerythrine SCHEMBL3319851 0.92 ALDH1A1 (0.98) ALDH1A1MAPTSMN1; SMN2HPGDKMT2A
Chelerythrine SCHEMBL4016265 0.92 ALDH1A1 (0.98) ALDH1A1MAPTSMN1; SMN2HPGDKMT2A
Chelerythrine SCHEMBL4980861 0.92 ALDH1A1 (0.98) ALDH1A1MAPTSMN1; SMN2HPGDKMT2A
Chelerythrine SCHEMBL288916 0.92 ALDH1A1 (0.98) ALDH1A1MAPTSMN1; SMN2HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113207893-B Degerming composition containing moroxydine hydrochloride and degerming agent 一力制药股份有限公司 2022-01-11 CN disclosed
CN-113207893-A Degerming composition containing moroxydine hydrochloride and degerming agent 一力制药股份有限公司 2021-08-06 CN disclosed