SCHEMBL28634720

SCHEMBL28634720

C=CCONC(=O)C(C)(C)Br

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.33
CACNA1B Q00975 1/20 0.33
APBA1 Q02410 1/20 0.33
CYP3A4 P08684 1/20 0.32
TSHR P16473 2/20 0.31
HSD17B10 Q99714 1/20 0.31
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31
ADRB3 P13945 1/20 0.31
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30
CCNA1 P78396 1/20 0.30
CDK5 Q00535 1/20 0.30
CDK5R1 Q15078 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15341473 0.75 ALOX15 (0.32) ALDH1A1
SCHEMBL3053229 0.73 SMN1; SMN2 (0.41) ALDH1A1MAPTCACNA1BAPBA1
SCHEMBL873545 0.73
SCHEMBL7564252 0.71 MAPT (0.34) ALDH1A1MAPTCACNA1BAPBA1TSHR
SCHEMBL694328 0.70
SCHEMBL873544 0.70
SCHEMBL1894433 0.70
SCHEMBL28510539 0.69
SCHEMBL463385 0.69 CYP3A4 (0.42) ALDH1A1MAPTCACNA1BAPBA1CYP3A4
SCHEMBL16265028 0.69 ALDH1A1 (0.38) ALDH1A1MAPTCYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429424-B Preparation method of [1,2,4] oxadiazino indoline-3-ketone derivative 华侨大学 2022-06-07 CN claimed
CN-113429424-A Preparation method of [1,2,4] oxadiazino indoline-3-ketone derivative 华侨大学 2021-09-24 CN claimed
CN-113429424-B Preparation method of [1,2,4] oxadiazino indoline-3-ketone derivative 华侨大学 2022-06-07 CN disclosed
CN-113429424-A Preparation method of [1,2,4] oxadiazino indoline-3-ketone derivative 华侨大学 2021-09-24 CN disclosed