SCHEMBL28636337

SCHEMBL28636337

CCc1nc2c(C)c(Cl)ccc2c(Nc2cccc(O)c2)c1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 1/20 0.41
TRPV1 Q8NER1 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
POLB P06746 1/20 0.39
RAD52 P43351 1/20 0.39
GFER P55789 1/20 0.39
PIM1 P11309 2/20 0.39
PIM2 Q9P1W9 1/20 0.39
MAPT P10636 4/20 0.38
CSNK2A1 P68400 2/20 0.38
FABP3 P05413 1/20 0.38
FABP4 P15090 1/20 0.38
FABP5 Q01469 1/20 0.38
CSNK2A2 P19784 1/20 0.38
CSNK2B P67870 1/20 0.38
TOP2A P11388 1/20 0.37
TP53 P04637 2/20 0.37
ALOX5 P09917 1/20 0.37
RAPGEF4 Q8WZA2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18292471 0.73 TP53 (0.67) POLBMAPTTP53GAAMAPK1
SCHEMBL5929645 0.65 FABP3 (0.47) PPARAMEN1KMT2ACSNK2A1FABP3
SCHEMBL3061423 0.65 DHODH (0.50) KMT2AFABP3FABP4FABP5TP53
SCHEMBL4433976 0.65 CSF1R (0.48) MAPTCSNK2A1FABP3FABP4FABP5
SCHEMBL3066041 0.63 DHODH (0.47) KMT2AFABP3FABP4FABP5
SCHEMBL28204900 0.62 FABP4 (0.46) MEN1KMT2AFABP3FABP4FABP5
SCHEMBL20138876 0.62 PDE10A (0.40) MEN1KMT2AMAPTFABP3FABP4
SCHEMBL1841268 0.62 P2RX3 (0.43) MAPT
SCHEMBL20138862 0.61 FABP4 (0.44) KMT2AFABP3FABP4FABP5GAA
SCHEMBL17060022 0.60 CYP3A4 (0.60) MEN1KMT2APOLBRAD52GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109730996-B Quinoline structure type androgen receptor antagonist and application thereof 浙江大学 2021-08-24 CN disclosed