SCHEMBL5929645

SCHEMBL5929645

CCc1nc2cc(Cl)c(Cl)cc2c(Nc2ccccc2C)c1C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FABP3 P05413 2/20 0.47
FABP4 P15090 2/20 0.47
FABP5 Q01469 1/20 0.47
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
PTGS2 P35354 1/20 0.41
FTO Q9C0B1 1/20 0.40
CYP2C9 P11712 1/20 0.40
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
PPARG P37231 1/20 0.40
RXRG P48443 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40
CSNK2A1 P68400 1/20 0.39
C1R P00736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6108087 0.73 CSF1R (0.53) CYP2C9
SCHEMBL5929643 0.71 MAPT (0.65)
SCHEMBL8569897 0.69 LMNA (0.43) MEN1KMT2A
SCHEMBL4433976 0.69 CSF1R (0.48) FABP3FABP4FABP5CSNK2A1
SCHEMBL6293298 0.68 FABP3 (0.61) FABP3FABP4FABP5MEN1KMT2A
Acetic Acid SCHEMBL21725059 0.67 PTGS2 (0.61) FABP3FABP4MEN1KMT2APTGS2
SCHEMBL6109140 0.66 FABP3 (0.40) FABP3FABP4FABP5MEN1KMT2A
SCHEMBL537930 0.65 FABP4 (0.46) FABP3FABP4FABP5MEN1KMT2A
SCHEMBL28636337 0.65 PPARA (0.41) FABP3FABP4FABP5MEN1KMT2A
SCHEMBL11545050 0.65 FABP4 (0.64) FABP3FABP4FABP5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060173034-A1 Novel 4-anilinoquinoline-3-carboxamides ASTRAZENECA AB (SE) 2006-08-03 US disclosed
US-7037925-B2 4-anilinoquinoline-3-carboxamides ASTRAZENECA AB (SE) 2006-05-02 US disclosed
EP-1387830-A1 NOVEL 4-ANILINOQUINOLINE-3-CARBOXAMIDES AstraZeneca AB (SE) 2004-02-11 EP disclosed
WO-2002092571-A1 NOVEL 4-ANILINOQUINOLINE-3-CARBOXAMIDES ASTRAZENECA AB (SE) 2002-11-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060173034-A1 Novel 4-anilinoquinoline-3-carboxamides JAK3, JAK2, JAK1 FABP3 2197/4885FABP4 3563/4885FABP5 3852/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.