SCHEMBL28636889

SCHEMBL28636889

FC(F)(F)c1ccc(N=c2[nH]c(-c3ccc(Br)cc3)cs2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.47
IDO1 P14902 1/20 0.44
AHR P35869 2/20 0.34
SCN2A Q99250 2/20 0.33
KIF11 P52732 2/20 0.33
CCNB2 O95067 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
MPI P34949 1/20 0.33
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
PLAU P00749 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28195676 0.88 MAPT (0.45) TRPV1SCN2AKIF11CCNB2CDK1
SCHEMBL28646823 0.86 ALDH1A1 (0.44) IDO1SCN2AKIF11CCNB2CDK1
SCHEMBL28195673 0.86 KIF11 (0.33) TRPV1SCN2AKIF11CCNB2CDK1
SCHEMBL28627573 0.86 MAPT (0.44) TRPV1IDO1SCN2AKIF11CCNB2
SCHEMBL28195733 0.86 GCGR (0.39) TRPV1IDO1SCN2AKIF11CCNB2
SCHEMBL28195066 0.86 SCN2A (0.43) IDO1SCN2AKIF11MPIALDH1A1
SCHEMBL28195679 0.85 IDO1 (0.35) TRPV1IDO1SCN2AKIF11MPI
SCHEMBL28195019 0.84 TRPA1 (0.38) TRPV1KIF11CCNB2CDK1CCNB1
SCHEMBL28195670 0.83 KIF11 (0.51) KIF11ALDH1A1MAPTGCGRMAPK14
SCHEMBL28195054 0.83 NPBWR1 (0.39) IDO1KIF11HTR3EHTR3BPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107629022-B Antibacterial synergist and preparation method and application thereof 上海医药工业研究院 2024-11-12 CN disclosed
CN-107625766-B Application of thiazole compound as antibacterial synergist 上海医药工业研究院 2021-08-31 CN disclosed
CN-107629023-A A kind of new fragrant imido grpup thiazole compound, preparation method and use 华东理工大学 2018-01-26 CN disclosed
CN-107625766-A A kind of thiazole compound is used as the purposes of Trimethoprim 上海医药工业研究院 2018-01-26 CN disclosed
CN-107629022-A A kind of Trimethoprim and its preparation method and purposes 上海医药工业研究院 2018-01-26 CN disclosed