SCHEMBL28637014

SCHEMBL28637014

CCCc1nc(-c2cccnc2N)n[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.41
MKNK1 Q9BUB5 2/20 0.38
MKNK2 Q9HBH9 2/20 0.38
CDK1 P06493 1/20 0.38
CDK2 P24941 1/20 0.38
RPS6KA5 O75582 1/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
NOS2 P35228 2/20 0.36
VCP P55072 1/20 0.36
HPGD P15428 1/20 0.36
PDPK1 O15530 1/20 0.36
MAP4K4 O95819 1/20 0.36
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
NFKB1 P19838 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12395279 0.71 S1PR1 (0.59) HPGDKDM4ENPC1HTTRAB9A
SCHEMBL29109555 0.69 DDX3X (0.40) AOC3KDM4ENPC1NFKB1HTT
SCHEMBL2384178 0.69 BACE1 (0.51) NOS2VCPKDM4ETDP1NOS3
SCHEMBL16432027 0.68 MAP4K4 (0.53) MKNK1MKNK2CDK1CDK2NOS2
SCHEMBL12474028 0.68 MKNK1 (0.51) MKNK1MKNK2RPS6KA5NOS2HPGD
SCHEMBL26108844 0.68 NR1H2 (0.50) NR1H2NR1H3KDM4ENPC1NFKB1
SCHEMBL31228708 0.68 NR1H2 (0.50) NR1H2NR1H3KDM4ENPC1NFKB1
SCHEMBL7324860 0.67 ALPL (0.46) MKNK1MKNK2CDK1CDK2HPGD
SCHEMBL7659462 0.67 DDX3X (0.43) NR1H2NR1H3TLR8ALPL
SCHEMBL27880002 0.67 SMN1; SMN2 (0.56) HPGDKDM4ENPC1NFKB1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113227070-A ASK1 inhibitors 比奥根MA公司 2021-08-06 CN disclosed