SCHEMBL28638166

SCHEMBL28638166

CCOc1cc2c(cc1C(=O)O)CN(C(C)c1ccccc1)C2=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
MAPK1 P28482 4/20 0.42
MAPT P10636 1/20 0.41
THRB P10828 2/20 0.40
GAA P10253 1/20 0.40
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
XIAP P98170 1/20 0.39
HKDC1 Q2TB90 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
NOD2 Q9HC29 1/20 0.39
MEN1 O00255 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28645332 0.91 LMNA (0.41) KMT2AMAPK1MAPTTHRBKDM4E
SCHEMBL28651754 0.80 KMT2A (0.49) KMT2AMAPTGAAKDM4EALOX15
SCHEMBL28633462 0.78 KMT2A (0.53) KMT2AMAPTALOX15TDP1MEN1
SCHEMBL28645763 0.77 KMT2A (0.41) KMT2AALOX15TSHRHSD17B10MEN1
SCHEMBL28652352 0.76 KMT2A (0.48) KMT2AKDM4EALDH1A1ALOX15TSHR
SCHEMBL28644854 0.76 KMT2A (0.48) KMT2AMAPTKDM4EALDH1A1TSHR
SCHEMBL30604559 0.76 KMT2A (0.48) KMT2AMAPTKDM4EALDH1A1TSHR
SCHEMBL28652153 0.73 KMT2A (0.53) KMT2AKDM4EMEN1TP53LMNA
SCHEMBL28645344 0.73 KMT2A (0.41) KMT2AKDM4EALOX15TSHRHSD17B10
SCHEMBL6288893 0.73 TP53 (0.53) KMT2AMAPTTHRBGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493438-A Tetrahydroisoquinoline compounds 江苏先声药业有限公司 2021-10-12 CN disclosed