SCHEMBL28645332

SCHEMBL28645332

CCOC(=O)c1cc2c(cc1OCC)C(=O)N(C(C)c1ccccc1)C2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.41
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
GABRA1 P14867 2/20 0.40
GABRB2 P47870 2/20 0.40
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSP90AA1 P07900 1/20 0.40
ABCB11 O95342 1/20 0.40
GABRA2 P47869 1/20 0.40
MAPK1 P28482 3/20 0.40
THRB P10828 2/20 0.40
MAPT P10636 3/20 0.39
TP53 P04637 2/20 0.39
ALDH1A1 P00352 2/20 0.39
POLB P06746 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28638166 0.91 KMT2A (0.46) LMNAMAPK1THRBMAPTTP53
SCHEMBL28925170 0.81 CASP3 (0.47) HSP90AA1MAPK1MAPTTP53ALDH1A1
SCHEMBL28639031 0.79 KMT2A (0.57) CYP3A4CYP2C9CYP2C19HSP90AA1ALDH1A1
SCHEMBL28656587 0.78 TSHR (0.51) HSP90AA1MAPTTP53MEN1KMT2A
SCHEMBL30604600 0.78 HSP90AA1 (0.43) HSP90AA1MAPTTP53ALDH1A1POLB
SCHEMBL28640895 0.78 HSP90AA1 (0.43) HSP90AA1MAPTTP53ALDH1A1POLB
SCHEMBL28645772 0.78 PARP1 (0.40) GABRA1HSP90AA1GABRA2MAPTTP53
SCHEMBL28633459 0.73 MEN1 (0.47) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL30604585 0.73 MEN1 (0.47) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL28926168 0.73 MEN1 (0.39) LMNACYP1A2GABRA1CYP2C19HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493438-B Tetrahydroisoquinoline compounds 南京再明医药有限公司 2023-10-20 CN disclosed
CN-113493438-A Tetrahydroisoquinoline compounds 江苏先声药业有限公司 2021-10-12 CN disclosed