SCHEMBL28639443

SCHEMBL28639443

CC1(C)OB(c2cc(C3CC3)nc3c2ccn3S(=O)(=O)Cc2ccccc2)OC1(C)C

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.33
DRD2 P14416 2/20 0.32
HTR6 P50406 2/20 0.32
SMYD3 Q9H7B4 2/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
POLB P06746 1/20 0.31
HSD17B10 Q99714 2/20 0.31
TSHR P16473 1/20 0.31
USP2 O75604 1/20 0.31
ATM Q13315 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28657466 0.85 CYP2C19 (0.41) CYP2C19DRD2HTR6MEN1KMT2A
SCHEMBL28639441 0.81 RAPGEF4 (0.33)
SCHEMBL20443037 0.72
SCHEMBL28802488 0.71 CYP2C19 (0.36) CYP2C19ALDH1A1
SCHEMBL23403834 0.69 PDE4A (0.35) CYP2C19ALDH1A1MAPTNPSR1
SCHEMBL28852707 0.69 HTR6 (0.36) CYP2C19HTR6TSHRALDH1A1HPGD
SCHEMBL29414040 0.69 HTR6 (0.36) CYP2C19HTR6TSHRALDH1A1HPGD
SCHEMBL28333115 0.68 DGAT1 (0.33) CYP2C19ALDH1A1
SCHEMBL28333074 0.68 ALDH1A1 (0.38) CYP2C19KMT2AHSD17B10TSHRALDH1A1
SCHEMBL28657465 0.66 RAPGEF4 (0.37) CYP2C19ALDH1A1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110198941-B Pyrrolopyridine N-oxide derivative and preparation method and application thereof 江苏豪森药业集团有限公司 2021-09-28 CN disclosed