SCHEMBL28644262

SCHEMBL28644262

CNc1ccc(S(=O)(=O)c2ccc(OC)cc2)s1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 5/20 0.59
LOX P28300 2/20 0.58
GAA P10253 1/20 0.51
CA2 P00918 3/20 0.51
CFTR P13569 1/20 0.44
MMP2 P08253 4/20 0.44
MMP8 P22894 4/20 0.44
MMP13 P45452 4/20 0.44
MMP9 P14780 3/20 0.44
MMP1 P03956 2/20 0.44
CA1 P00915 1/20 0.44
RAPGEF4 Q8WZA2 1/20 0.43
HSD11B1 P28845 1/20 0.42
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.40
MMP12 P39900 3/20 0.40
MMP14 P50281 3/20 0.40
MMP16 P51512 3/20 0.40
MMP3 P08254 1/20 0.40
ADAM17 P78536 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28651581 0.82 LOX (0.53) LOXHSD11B1ALDH1A1HPGD
SCHEMBL28645837 0.82 LOX (0.55) LOXGAA
SCHEMBL14486413 0.77 PKM (1.00) PKMLOXGAACA2MMP2
SCHEMBL13074716 0.77 PKM (1.00) PKMLOXGAACA2MMP2
SCHEMBL835692 0.77 PKM (1.00) PKMLOXGAACA2MMP2
Hydrochloric Acid SCHEMBL28644204 0.77 LOX (0.55) LOXCA2MMP2MMP8MMP13
Hydrochloric Acid SCHEMBL28661275 0.76 LOXL2 (0.67) LOX
SCHEMBL28156749 0.76 CFTR (0.47) PKMLOXGAACA2CFTR
SCHEMBL28646901 0.76 LOXL2 (0.58) PKMLOX
SCHEMBL19259654 0.75 PKM (0.59) PKMLOXGAACA2CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311839-B Methylamine derivatives as lysyl oxidase inhibitors for the treatment of cancer 癌症研究协会皇家癌症医院 2021-11-02 CN disclosed