SCHEMBL28644286

SCHEMBL28644286

NC(=O)OCc1ncc(Sc2cc3ccccc3c3ccccc23)s1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 6/20 0.41
MAOA P21397 2/20 0.41
NTRK1 P04629 1/20 0.33
SIRT2 Q8IXJ6 5/20 0.33
LOXL3 P58215 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
SIRT3 Q9NTG7 1/20 0.33
ICAM1 P05362 4/20 0.32
SELE P16581 4/20 0.32
VCAM1 P19320 1/20 0.32
HTT P42858 2/20 0.32
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2C19 P33261 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LOX P28300 1/20 0.31
KCNH2 Q12809 1/20 0.31
AOC3 Q16853 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28651627 0.87 SIRT2 (0.43) LOXL2SIRT2SIRT1SIRT3HTT
SCHEMBL28663602 0.82 SIRT2 (0.44) LOXL2NTRK1SIRT2LOXL3SIRT1
SCHEMBL28644238 0.79 LOXL2 (0.41) LOXL2NTRK1LOXL3SIRT1ICAM1
SCHEMBL19259879 0.78 LOXL2 (0.39) LOXL2MAOANTRK1SIRT2LOXL3
SCHEMBL28657391 0.76 LOXL2 (0.43) LOXL2NTRK1SIRT2LOXL3SIRT1
SCHEMBL19274717 0.75 PDPK1 (0.44) LOXL2MAOACYP1A2
SCHEMBL28644194 0.74 LOXL2 (0.42) LOXL2NTRK1LOXL3HTTALDH1A1
SCHEMBL28643885 0.73 LOXL3 (0.36) LOXL2NTRK1LOXL3ICAM1SELE
SCHEMBL28645865 0.72 LOXL2 (0.40) LOXL2NTRK1LOXL3ICAM1SELE
SCHEMBL28651596 0.71 ALDH1A1 (0.42) LOXL2LOXL3ICAM1SELEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311839-B Methylamine derivatives as lysyl oxidase inhibitors for the treatment of cancer 癌症研究协会皇家癌症医院 2021-11-02 CN disclosed